SCHEMBL5050844

SCHEMBL5050844

CC(=O)OCCN(CCO)CCNC(=O)c1ccc(CN)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.45
LMNA P02545 2/20 0.45
SLC22A2 O15244 1/20 0.45
SLC22A1 O15245 1/20 0.45
TSHR P16473 1/20 0.45
ACHE P22303 1/20 0.45
MAPK1 P28482 1/20 0.45
CYP2C19 P33261 1/20 0.45
BLM P54132 2/20 0.44
PMP22 Q01453 1/20 0.44
NFKB1 P19838 1/20 0.43
KCNH2 Q12809 1/20 0.43
POLB P06746 3/20 0.42
CYP3A4 P08684 2/20 0.42
MCHR1 Q99705 1/20 0.42
THRB P10828 1/20 0.42
ATM Q13315 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
HDAC3 O15379 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5050842 0.88 ALDH1A1 (0.47) ALDH1A1LMNASLC22A2SLC22A1TSHR
SCHEMBL8404683 0.88 LMNA (0.52) ALDH1A1LMNASLC22A2SLC22A1TSHR
SCHEMBL5008266 0.83 ALDH1A1 (0.51) ALDH1A1LMNASLC22A2SLC22A1TSHR
SCHEMBL19634682 0.82 KMT2A (0.55) ALDH1A1TSHRNFKB1CYP3A4MCHR1
SCHEMBL8404684 0.77 ALDH1A1 (0.56) ALDH1A1LMNASLC22A2SLC22A1TSHR
SCHEMBL19634425 0.77 ALDH1A1 (0.73) ALDH1A1LMNASLC22A2SLC22A1TSHR
SCHEMBL15947383 0.75 ALDH1A1 (0.50) ALDH1A1LMNASLC22A2SLC22A1TSHR
SCHEMBL5009757 0.74 ALDH1A1 (0.60) ALDH1A1LMNASLC22A2SLC22A1TSHR
SCHEMBL8404664 0.73 HDAC3 (0.61) TSHRBLMPMP22NFKB1POLB
SCHEMBL13496897 0.73 LMNA (0.48) ALDH1A1LMNASLC22A2SLC22A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1884513-A1 PYRAZOLE COMPOUND AND THERAPEUTIC AGENT FOR DIABETES COMPRISING THE SAME Japan Tobacco, Inc. (JP) 2008-02-06 EP disclosed