SCHEMBL5077508

SCHEMBL5077508

CC(C)(C)[SiH2]O[C]1C=Cc2ccccc21

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.34
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
ALDH1A1 P00352 2/20 0.34
HSD17B10 Q99714 2/20 0.34
MAPT P10636 2/20 0.34
ALOX15 P16050 2/20 0.34
KDM4E B2RXH2 1/20 0.34
BCHE P06276 1/20 0.34
POLB P06746 1/20 0.34
PTPRC P08575 1/20 0.34
THRB P10828 1/20 0.34
PKM P14618 1/20 0.34
IDO1 P14902 1/20 0.34
HPGD P15428 1/20 0.34
PTPN1 P18031 1/20 0.34
ACHE P22303 1/20 0.34
CES1 P23141 1/20 0.34
RECQL P46063 1/20 0.34
PTPN22 Q9Y2R2 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL756302 0.71 LMNA (0.41) LMNAMEN1KMT2AALDH1A1HSD17B10
SCHEMBL5077511 0.69
SCHEMBL7944967 0.69 SETD7 (0.37) LMNAMEN1KMT2AALDH1A1HSD17B10
SCHEMBL7635858 0.69 LMNA (0.33) LMNAMEN1KMT2AALDH1A1HSD17B10
SCHEMBL5693109 0.67 LMNA (0.41) LMNAMEN1KMT2AALDH1A1HSD17B10
SCHEMBL217367 0.67 LMNA (0.38) LMNAMEN1KMT2AALDH1A1HSD17B10
SCHEMBL705016 0.65 CA4 (0.42) LMNAALDH1A1ALOX15HPGDCYP2D6
SCHEMBL10435815 0.64 SETD7 (0.37) LMNAMEN1KMT2AALDH1A1HSD17B10
SCHEMBL1030000 0.63 LMNA (0.41) LMNAMEN1KMT2AALDH1A1HSD17B10
SCHEMBL3769766 0.62 MEN1 (0.55) LMNAMEN1KMT2AALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001070395-A2 POLYMERIZATION CATALYSTS COMPRISING AN OPEN ETA-5 LIGAND BOREALIS TECHNOLOGY OY (FI) 2001-09-27 WO claimed
EP-1412392-B1 METALLOCENE CATALYST CONTAINING A CYCLOPENTADIENYL LIGAND SUBSTITUTED BY A SILOXY OR GERMYLOXY GROUP CONTAINING AN OLEFINIC RESIDUE BOREALIS TECH OY (FI) 2008-03-26 EP disclosed
US-7037872-B2 Metallocene catalysts containing a cyclopentadienyl ligand substituted by a siloxy or germiloxy group containing an olefinic residue BOREALIS TECHNOLOGY OY (FI) 2006-05-02 US disclosed
US-20040198590-A1 Metallocene catalysts containing a cyclopentadienyl ligand substituted by a siloxy or germiloxy group containing an olefinic residue BOREALIS TECHNOLOGY OY (FI) 2004-10-07 US disclosed
EP-1412392-A1 METALLOCENE CATALYST CONTAINING A CYCLOPENTADIENYL LIGAND SUBSTITUTED BY A SILOXY OR GERMYLOXY GROUP CONTAINING AN OLEFINIC RESIDUE Borealis Technology Oy (FI) 2004-04-28 EP disclosed
EP-1401880-A1 METALLOCENE CATALYSTS CONTAINING AN INDENYL MOIETY SUBSTITUTED AT THE 4-, 5-, 6- OR 7-POSITION BY A SILOXY OR GERMYLOXY GROUP Borealis Technology Oy (FI) 2004-03-31 EP disclosed
WO-2003010208-A1 METALLOCENE CATALYSTS CONTAINING A CYCLOPENTADIENYL LIGAND SUBSTITUTED BY A SILOXY OR GERMILOXY GROUP CONTAINING AN OLEFINIC RESIDUE BOREALIS TECHNOLOGY OY (FI) 2003-02-06 WO disclosed
WO-2003000744-A1 METALLOCENE CATALYSTS CONTAINING AN IDENYL MOIETY SUBSTITUTED AT THE 4-, 5-, 6- OR 7-POSITION BY A SILOXY OR GERMYLOXY GROUP BOREALIS TECHNOLOGY OY (FI) 2003-01-03 WO disclosed
EP-1248806-A1 METALLOCENE CATALYSTS COMPRISING MONOCYCLIC SILOXY SUBSTITUTED CYCLOPENTADIENYL GROUP(S) FOR THE POLYMERISATION OF OLEFINS Borealis Technology Oy (FI) 2002-10-16 EP disclosed
WO-2001070395-A2 POLYMERIZATION CATALYSTS COMPRISING AN OPEN ETA-5 LIGAND BOREALIS TECHNOLOGY OY (FI) 2001-09-27 WO disclosed
WO-2001053361-A1 SILOXY-SUBSTITUTED MONOCYCLOPENTADIENYL LIGATED CONSTRAINED GEOMETRY OLEFIN POLYMERISATION CATALYSTS BOREALIS TECHNOLOGY OY (FI) 2001-07-26 WO disclosed
WO-2001053362-A1 METALLOCENE CATALYSTS COMPRISING MONOCYCLIC SILOXY SUBSTITUTED CYCLOPENTADIENYL GROUP(S) FOR THE POLYMERISATION OF OLEFINS BOREALIS TECHNOLOGY OY (FI) 2001-07-26 WO disclosed