SCHEMBL508229

SCHEMBL508229

Cc1cc(N)ccc1OCC(C)(C)CO

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NUDT1 P36639 5/20 0.47
VDR P11473 6/20 0.40
PDE10A Q9Y233 1/20 0.39
ALDH1A1 P00352 3/20 0.38
PIM1 P11309 2/20 0.37
PIM2 Q9P1W9 2/20 0.37
AAK1 Q2M2I8 1/20 0.36
HDAC3 O15379 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
GAA P10253 3/20 0.36
KDM4E B2RXH2 2/20 0.36
MAPT P10636 2/20 0.36
MEN1 O00255 1/20 0.36
USP2 O75604 1/20 0.36
TP53 P04637 1/20 0.36
POLB P06746 1/20 0.36
CASP1 P29466 1/20 0.36
HTT P42858 1/20 0.36
CASP7 P55210 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8175332 0.90 ALDH1A1 (0.43) VDRPDE10AALDH1A1AAK1HDAC3
SCHEMBL942491 0.83 VDR (0.51) VDRPDE10AALDH1A1HDAC3HDAC6
SCHEMBL13723909 0.83 GAA (0.57) NUDT1ALDH1A1GAAKDM4EMAPT
SCHEMBL14320713 0.81 GAA (0.55) NUDT1ALDH1A1GAAKDM4EMAPT
SCHEMBL5857533 0.79 KDM4E (0.54) NUDT1ALDH1A1AAK1KDM4EUSP2
SCHEMBL2565945 0.78 ALDH1A1 (0.52) PDE10AALDH1A1AAK1GAAKDM4E
Hydrochloric Acid SCHEMBL5859058 0.78 KDM4E (0.53) NUDT1ALDH1A1AAK1KDM4EUSP2
SCHEMBL11704652 0.76 KDM4E (0.47) PDE10AALDH1A1GAAKDM4EMAPT
SCHEMBL9853450 0.75 KDM4E (0.37) VDRALDH1A1AAK1HDAC3HDAC6
SCHEMBL20496733 0.75 ALDH1A1 (0.50) PDE10AALDH1A1GAAKDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8580780-B2 6 substituted 2, 3,4,5 tetrahydro-1H-benzo[d]azepines as 5-HT2C receptor agonist ELI LILLY AND COMPANY (US) 2013-11-12 US disclosed
US-20120028961-A1 6 Substituted 2, 3,4,5 Tetrahydro-1H-Benzo[d]Azepines as 5-HT2c Receptor Agonist ELI LILLY AND COMPANY (US) 2012-02-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120028961-A1 6 Substituted 2, 3,4,5 Tetrahydro-1H-Benzo[d]Azepines as 5-HT2c Receptor Agonist HTR2C, HTR4, HTR1A NUDT1 3876/4885VDR 620/4885PDE10A 1911/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.