SCHEMBL509519

SCHEMBL509519

[NH]C(=O)CCSSc1ccccn1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.55
EHMT2 Q96KQ7 1/20 0.50
EHMT1 Q9H9B1 1/20 0.50
APOBEC3G Q9HC16 1/20 0.50
MAPT P10636 3/20 0.48
KMT2A Q03164 2/20 0.48
POLB P06746 2/20 0.47
MEN1 O00255 1/20 0.41
PKM P14618 1/20 0.41
NPC1 O15118 6/20 0.41
RAB9A P51151 6/20 0.41
SMN1; SMN2 Q16637 6/20 0.41
HPGD P15428 5/20 0.41
LMNA P02545 1/20 0.40
HDAC1 Q13547 1/20 0.39
HDAC2 Q92769 1/20 0.39
HSD17B10 Q99714 2/20 0.39
KDM4E B2RXH2 1/20 0.39
ALOX15 P16050 1/20 0.39
TDP1 Q9NUW8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL98030 0.87 ALDH1A1 (0.73) ALDH1A1EHMT2EHMT1APOBEC3GMAPT
SCHEMBL29811281 0.87 ALDH1A1 (0.73) ALDH1A1EHMT2EHMT1APOBEC3GMAPT
SCHEMBL8681802 0.85 ALDH1A1 (0.57) ALDH1A1EHMT2EHMT1APOBEC3GMAPT
SCHEMBL30308346 0.85 ALDH1A1 (0.71) ALDH1A1EHMT2EHMT1APOBEC3GMAPT
Succinic Acid SCHEMBL28529727 0.85 ALDH1A1 (0.71) ALDH1A1EHMT2EHMT1APOBEC3GMAPT
SCHEMBL13739021 0.85 ALDH1A1 (0.57) ALDH1A1EHMT2EHMT1APOBEC3GMAPT
SCHEMBL76157 0.84 ALDH1A1 (0.55) ALDH1A1EHMT2EHMT1APOBEC3GMAPT
SCHEMBL10064444 0.84 ALDH1A1 (0.55) ALDH1A1EHMT2EHMT1APOBEC3GMAPT
SCHEMBL18519250 0.84 ALDH1A1 (0.55) ALDH1A1EHMT2EHMT1APOBEC3GMAPT
SCHEMBL123215 0.83 ALDH1A1 (0.62) ALDH1A1EHMT2EHMT1APOBEC3GMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 191 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240238432-A1 METHOD FOR GLYCOPROTEIN MODIFICATION HONEYBEAR BIOSCIENCES INC. (TW) 2024-07-18 US claimed
WO-2024145600-A1 METHOD FOR GLYCOPROTEIN MODIFICATION HONEYBEAR BIOSCIENCES INC. (TW) 2024-07-04 WO claimed
CN-110914259-A Novel water-soluble mono-and di-branched complexing agents and corresponding lanthanide complexes CISBIO生物试验公司 2020-03-24 CN claimed
US-20090098574-A1 FUNCTIONALIZATION OF GOLD NANOPARTICLES WITH ORIENTED PROTEINS, APPLICATION TO THE HIGH-DENSITY LABELLING OF CELL MEMBRANES CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (CNRS) 2009-04-16 US claimed
EP-2018559-A1 FUNCTIONALIZATION OF GOLD NANOPARTICLES WITH ORIENTED PROTEINS. APPLICATION TO THE HIGH-DENSITY LABELLING OF CELL MEMBRANES Centre National de la Recherche Scientifique (CNRS) (FR) 2009-01-28 EP claimed
WO-2007122259-A1 FUNCTIONALIZATION OF GOLD NANOPARTICLES WITH ORIENTED PROTEINS. APPLICATION TO THE HIGH-DENSITY LABELLING OF CELL MEMBRANES CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (CNRS) (FR) 2007-11-01 WO claimed
US-20240238432-A1 METHOD FOR GLYCOPROTEIN MODIFICATION HONEYBEAR BIOSCIENCES INC. (TW) 2024-07-18 US disclosed
US-20240226322-A1 FIBRIN-SPECIFIC MATERIALS AND METHODS OF USING THEREOF NORTH CAROLINA STATE UNIVERSITY 2024-07-11 US disclosed
WO-2024145600-A1 METHOD FOR GLYCOPROTEIN MODIFICATION HONEYBEAR BIOSCIENCES INC. (TW) 2024-07-04 WO disclosed
US-11987558-B1 ALK5 inhibitors and their uses SYNTHIS THERAPEUTICS, INC. (US) 2024-05-21 US disclosed
US-20230295338-A1 A NOVEL ANTIBODY BINDING SPECIFICALLY TO HUMAN CEACAM1/3/5 AND USE THEREOF YMMUNOBIO AG (CH) 2023-09-21 US disclosed
US-20230132568-A1 ANTIBODY-ALK5 INHIBITOR CONJUGATES AND THEIR USES SYNTHIS THERAPEUTICS, INC. (US) 2023-05-04 US disclosed
US-20230090552-A1 ALK5 INHIBITOR CONJUGATES AND USES THEREOF SYNTHIS THERAPEUTICS, INC. (US) 2023-03-23 US disclosed
US-6197299-B1 TARGET CELL IS CONTACTED WITH A TARGET CELL LYSIS EFFECTIVE AMOUNT OF A SOLUBLE MONOCLONAL ANTIBODY OR FRAGMENT CONJUGATE COVALENTLY LINKED BY PEPTIDE BOND LINKAGE TO A SUPERANTIGEN FOR THE LYSIS OF A TARGET CELL BY ASSISTANCE OF LYMPHOCYTES PHARMACIA & UPJOHN AB (SE) 2001-03-06 US disclosed
WO-1999013918-A2 ICAM-1 SELECTIVE ECHOGENIC MICROBUBBLES UNIVERSITY OF PITTSBURGH (US) 1999-03-25 WO disclosed
EP-0610179-B1 TARGET SPECIFIC ANTIBODY-SUPERANTIGEN CONJUGATES AND THEIR PREPARATION PHARMACIA AB (SE) 1996-10-16 EP disclosed
EP-0610179-A1 TARGET SPECIFIC ANTIBODY-SUPERANTIGEN CONJUGATES AND THEIR PREPARATION. KABI PHARMACIA AB (SE) 1994-08-17 EP disclosed
EP-0540612-A1 HETEROBIFUNCTIONAL REAGENTS AND CONJUGATES WITH OXAALKYLENE UNITS FOR AMPHIPHILIC BRIDGE STRUCTURES Pharmacia AB (SE) 1993-05-12 EP disclosed
WO-1992001470-A1 TARGET SPECIFIC ANTIBODY-SUPERANTIGEN CONJUGATES AND THEIR PREPARATION KABI PHARMACIA AB (SE) 1992-02-06 WO disclosed
WO-1992001474-A1 HETEROBIFUNCTIONAL REAGENTS AND CONJUGATES WITH OXAALKYLENE UNITS FOR AMPHIPHILIC BRIDGE STRUCTURES KABI PHARMACIA AB (SE) 1992-02-06 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11987558-B1 ALK5 inhibitors and their uses ALK, ALKBH3, ALKBH5 ALDH1A1 1041/4885EHMT2 605/4885EHMT1 787/4885
US-20240238432-A1 METHOD FOR GLYCOPROTEIN MODIFICATION SIGLEC7, FUT5, FUT6 ALDH1A1 549/4885EHMT2 2301/4885EHMT1 2800/4885
US-20230090552-A1 ALK5 INHIBITOR CONJUGATES AND USES THEREOF ALK, ALKBH5, ALKBH3 ALDH1A1 297/4885EHMT2 268/4885EHMT1 260/4885
US-20230132568-A1 ANTIBODY-ALK5 INHIBITOR CONJUGATES AND THEIR USES ALK, ALKBH5, ALKBH3 ALDH1A1 346/4885EHMT2 468/4885EHMT1 629/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.