SCHEMBL51141

SCHEMBL51141

NS(=O)(=O)c1ncccn1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 11/20 0.43
CA2 P00918 11/20 0.43
CA9 Q16790 8/20 0.43
MAPK1 P28482 1/20 0.43
FTO Q9C0B1 1/20 0.39
HSP90AA1 P07900 1/20 0.38
CA12 O43570 7/20 0.38
CA6 P23280 4/20 0.38
CA7 P43166 3/20 0.38
CA13 Q8N1Q1 3/20 0.38
CA4 P22748 3/20 0.38
CA5A P35218 2/20 0.38
CA14 Q9ULX7 2/20 0.38
CA3 P07451 1/20 0.38
PLA2G7 Q13093 1/20 0.38
CA5B Q9Y2D0 1/20 0.38
LMNA P02545 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31527702 0.97 CA2 (0.42) CA1CA2CA9MAPK1FTO
Trimethylammonium SCHEMBL27851715 0.90 CA2 (0.38) CA1CA2CA9MAPK1FTO
Pyridine SCHEMBL9838377 0.88 NAPRT (0.41) CA1CA2CA9MAPK1FTO
Pyrrole SCHEMBL27616550 0.86 CA2 (0.36) CA1CA2CA9MAPK1FTO
Pyrazole SCHEMBL27514785 0.81 CA1 (0.33) CA1CA2CA9MAPK1FTO
Trifluoroacetic Acid SCHEMBL28163458 0.81 L3MBTL1 (0.41) CA1CA2CA9MAPK1FTO
SCHEMBL28576 0.79 CA1 (0.33) CA1CA2CA9MAPK1FTO
Imidazole SCHEMBL8354987 0.79 ALDH1A1 (0.48) CA1CA2CA9MAPK1FTO
1,2,4-Triazole SCHEMBL6053442 0.78 CA1 (0.32) CA1CA2CA9MAPK1CYP1A2
SCHEMBL5593062 0.75 TXNRD1 (0.37) CA1CA2CA9MAPK1HSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 664 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025102245-A1 SYNTHESIS METHOD FOR DUAL ENDOTHELIN RECEPTOR ANTAGONIST APROCITENTAN 浙江天宇药业股份有限公司 2025-05-22 WO claimed
CN-117736152-A Synthesis method of dual endothelin receptor antagonist apixitan 浙江天宇药业股份有限公司 2024-03-22 CN claimed
EP-3860998-B1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH APJ RECEPTOR ACTIVITY ANNAPURNA BIO INC (US) 2023-12-27 EP claimed
CN-109633065-B Method for detecting drug residues in animal body 沈阳海关技术中心 2021-04-20 CN claimed
EP-3255043-B1 N-(6-((2R,3S)-3,4-DIHYDROXYBUTAN-2-YLOXY)-2-(4-FLUOROBENZYLTHIO)PYRIMIDIN-4-YL)-3- METHYLAZETIDINE-1-SULFONAMIDE AS CHEMOKINE RECEPTOR MODULATOR ASTRAZENECA AB (SE) 2021-01-20 EP claimed
US-9975881-B2 Compound ASTRAZENECA AB (SE) 2018-05-22 US claimed
US-20160108023-A1 Novel Compound ASTRAZENECA AB (SE) 2016-04-21 US claimed
CN-103781781-B N-(6-((2R, 3S)-3,4-dihydroxyl fourth-2-base oxygen base)-2-(4-Fluorobenzylthio) pyrimidine-4-yl as chemokine receptor modulators)-3-methyl azetidine-1-sulphonamide ASTRAZENECA AB (SE) 2015-08-26 CN claimed
US-20140228339-A1 Novel Compound ASTRAZENECA AB (SE) 2014-08-14 US claimed
US-8735413-B2 Compound ASTRAZENECA AB (SE) 2014-05-27 US claimed
CN-1081815-A Safe with pyrazolyl sulfonylureas of activity of weeding MONSANTO CO (US) 1994-02-16 CN claimed
CN-1075846-A Chemically stabilized herbicidal oil-based suspensions ISHIHARA SANGYO KAISHA (JP) 1993-09-08 CN claimed
CN-1068824-A N-pyrazolyl-1, 2, 4-triazolo [1, 5-c ] pyrimidine-2-sulfonamides as herbicides DOWELANCO (US) 1993-02-10 CN claimed
CN-1063015-A Safe herbicidal sulfonamide compositions MONSANTO CO (US) 1992-07-29 CN claimed
CN-1054251-A 5,7-dihydroxyl-1,2, the preparation method of 4-triazolo [1,5-a] pyrimidine-2-sulfonanilide DOWELANCO (US) 1991-09-04 CN claimed
CN-1051561-A Preparation 5-methyl-N-aryl-1,2, the aqueous process of 4-triazolo [1,5-a] pyrimidine-2-sulfonamides DOWELANCO (US) 1991-05-22 CN claimed
EP-0142152-B1 Novel substituted 1,2,4-triazolo- [1,5-a] pyrimidine-2-sulfonamides and compositions and methods of controlling undesired vegetation and suppressing the nitrification of ammonium nitrogen in soil THE DOW CHEMICAL COMPANY (US) 1991-03-20 EP claimed
EP-0343752-A1 Alkoxy-1,2,4-triazolo (1,5-c) pyrimidine-2-sulfonamides, process for their preparation and intermediates DowElanco (US) 1989-11-29 EP claimed
EP-0337947-A1 Triazolylsulfonamides CIBA-GEIGY AG (CH) 1989-10-18 EP claimed
CN-1031174-A Herbicidal combinations ISHIHARA SANGYO KAISHA (JP) 1989-02-22 CN claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140228339-A1 Novel Compound CXCR2, CXCR1, CCR5 CA1 3867/4885CA2 2395/4885CA9 2447/4885
US-20160108023-A1 Novel Compound CXCR2, CXCR1, CCR5 CA1 3867/4885CA2 2395/4885CA9 2447/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.