Formamide

Formamide

SCHEMBL5126384

COc1ccc(N2CCC3(CC2)CC(C(=O)NN2CCN(c4ncccc4Cl)CC2)=NO3)cc1.NC=O

nearest known ligand 0.41

Full drug profile on Sugi Atlas →

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.41
ALDH1A1 P00352 2/20 0.41
TRPA1 O75762 5/20 0.40
TRPV1 Q8NER1 1/20 0.39
MALT1 Q9UDY8 2/20 0.39
LMNA P02545 1/20 0.37
TP53 P04637 1/20 0.37
RBP4 P02753 1/20 0.37
DRD2 P14416 1/20 0.37
HTR2A P28223 1/20 0.37
DGAT1 O75907 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
RAB9A P51151 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Formamide SCHEMBL5116397 0.88 DRD2 (0.38) MAPTTRPA1TRPV1MALT1DRD2
SCHEMBL1457231 0.85 TRPV1 (0.50) TRPA1TRPV1RBP4L3MBTL1
Formamide SCHEMBL5122603 0.80 CXCR3 (0.40) TRPV1L3MBTL1KMT2A
SCHEMBL5127608 0.74 TRPV1 (0.54) TRPA1TRPV1RBP4
SCHEMBL1457235 0.74 TRPV1 (0.48) TRPA1TRPV1MALT1
SCHEMBL1457227 0.73 P2RY12 (0.45) TRPA1TRPV1LMNAKMT2A
SCHEMBL5117962 0.73 P2RY12 (0.51) TRPA1TRPV1RBP4
SCHEMBL1457447 0.73 TRPA1 (0.45) TRPA1TRPV1MALT1RBP4
SCHEMBL1457424 0.71 TRPA1 (0.43) ALDH1A1TRPA1TRPV1MALT1RBP4
SCHEMBL5127551 0.70 RBP4 (0.62) TRPA1TRPV1MALT1RBP4KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080214807-A1 Substituted Spiro Compounds and their Use for Producing Drugs GRUENENTHAL GMBH (DE) 2008-09-04 US claimed
US-20080214807-A1 Substituted Spiro Compounds and their Use for Producing Drugs GRUENENTHAL GMBH (DE) 2008-09-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080214807-A1 Substituted Spiro Compounds and their Use for Producing Drugs REN, PKD1, NR3C2 MAPT 3811/4885ALDH1A1 281/4885TRPA1 720/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.