SCHEMBL5129072

SCHEMBL5129072

Cc1cc(CO)c(O)c(-c2cccc3ccccc23)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
PDCD1 Q15116 1/20 0.40
CD274 Q9NZQ7 1/20 0.40
MAOA P21397 1/20 0.40
MAOB P27338 1/20 0.40
IDH1 O75874 1/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
PTGS1 P23219 1/20 0.37
PTGS2 P35354 1/20 0.37
KDM4E B2RXH2 2/20 0.37
MAPT P10636 2/20 0.37
CYP1A2 P05177 2/20 0.37
CYP2A6 P11509 2/20 0.37
ALDH1A1 P00352 2/20 0.37
HPGD P15428 1/20 0.37
MPI P34949 1/20 0.37
MCL1 Q07820 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3680169 0.87 MAOA (0.45) MAOAMAOBMEN1KMT2APTGS1
SCHEMBL10089370 0.84 BCHE (0.44) CYP3A4CYP2C9CYP2C19MAOAMAOB
SCHEMBL10089369 0.83 EGFR (0.39) CYP3A4CYP2C9CYP2C19MAOAMAOB
SCHEMBL13044875 0.83 F2 (0.42) MAOAMAOBPTGS1PTGS2KDM4E
SCHEMBL17500079 0.82 CYP1A2 (0.48) MAOAMAOBPTGS1PTGS2KDM4E
SCHEMBL2331853 0.81 CYP2D6 (0.38) CYP2C9CYP2C19MEN1KMT2ACYP1A2
SCHEMBL10014387 0.78 PDCD1 (0.50) PDCD1CD274PTGS1ALDH1A1
SCHEMBL12445306 0.77 DHFR (0.35) CYP3A4CYP2C9CYP2C19PDCD1CD274
SCHEMBL17500089 0.77 SMN1; SMN2 (0.50) CYP2C9CYP2C19MAOAMAOBPTGS1
SCHEMBL13508862 0.77 HTR7 (0.38) CYP3A4CYP2C9CYP2C19MAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1973655-A2 POLYDENTATE HETEROATOM LIGAND CONTAINING METAL COMPLEXES, CATALYSTS AND METHODS OF MAKING AND USING THE SAME DOW GLOBAL TECHNOLOGIES INC. (US) 2008-10-01 EP disclosed
WO-2007075299-A2 POLYDENTATE HETEROATOM LIGAND CONTAINING METAL COMPLEXES, CATALYSTS AND METHODS OF MAKING AND USING THE SAME DOW GLOBAL TECHNOLOGIES INC. (US) 2007-07-05 WO disclosed