SCHEMBL5134741

SCHEMBL5134741

Cc1ccccc1OC1=CC(=O)C(N)=C(c2ncnc3ccccc23)C1=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 1/20 0.39
RAB9A P51151 3/20 0.37
USP2 O75604 1/20 0.37
SMN1; SMN2 Q16637 3/20 0.37
ADORA2A P29274 2/20 0.35
PKM P14618 1/20 0.35
PI4KA P42356 1/20 0.34
PI4K2B Q8TCG2 1/20 0.34
PI4K2A Q9BTU6 1/20 0.34
PI4KB Q9UBF8 1/20 0.34
CYP1A2 P05177 2/20 0.34
CYP2C19 P33261 2/20 0.34
MRGPRX1 Q96LB2 2/20 0.34
HSD17B10 Q99714 1/20 0.32
MAPT P10636 3/20 0.32
NPC1 O15118 2/20 0.32
ALDH1A1 P00352 2/20 0.32
LMNA P02545 1/20 0.32
HSP90AA1 P07900 1/20 0.32
XBP1 P17861 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5134739 0.92 MAP4K4 (0.40) MAP4K4RAB9AUSP2SMN1; SMN2ADORA2A
SCHEMBL5135030 0.84 GAPDH (0.42) MAP4K4RAB9AADORA2API4KAPI4K2B
SCHEMBL5135024 0.80 ADORA2A (0.43) RAB9AUSP2SMN1; SMN2ADORA2APKM
SCHEMBL5664809 0.79 LDHA (0.40) RAB9AADORA2API4KAPI4K2BPI4K2A
SCHEMBL5135022 0.74 ADORA2A (0.44) RAB9AUSP2SMN1; SMN2ADORA2APKM
SCHEMBL5135370 0.69 CES1 (0.47) RAB9ASMN1; SMN2ADORA2ANPC1HTT
SCHEMBL4364907 0.68 CYP1A2 (0.59) MAP4K4RAB9ASMN1; SMN2PI4KAPI4K2B
SCHEMBL5664944 0.65 KDR (0.43) TDP2NSD2PAX8HKDC1ATG4B
SCHEMBL5135297 0.64 APAF1 (0.43) MAP4K4ADORA2API4KAPI4K2BPI4K2A
SCHEMBL29049141 0.63 ADORA2A (0.46) RAB9AADORA2APKMPI4KAPI4K2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080268460-A1 Assays to Identify Irreversibly Binding Inhibitors of Receptor Tyrosine Kinases WYETH (US) 2008-10-30 US disclosed