SCHEMBL5137147

SCHEMBL5137147

FC(F)(F)c1cc(Cn2c[c]c3ccccc32)cc(C(F)(F)F)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.39
HTT P42858 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
IDO1 P14902 2/20 0.37
MAPT P10636 3/20 0.36
LMNA P02545 1/20 0.36
TP53 P04637 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
SIRT2 Q8IXJ6 1/20 0.35
SIRT1 Q96EB6 1/20 0.35
ICMT O60725 2/20 0.34
ALDH1A1 P00352 2/20 0.34
GAA P10253 2/20 0.34
TACR1 P25103 4/20 0.34
CACNA1F O60840 1/20 0.34
CACNA1D Q01668 1/20 0.34
CACNA1S Q13698 1/20 0.34
CACNA1C Q13936 1/20 0.34
TSHR P16473 1/20 0.34
HTR6 P50406 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5138333 0.87 HTR6 (0.45) KDM4ESMN1; SMN2IDO1MAPTLMNA
SCHEMBL4600343 0.80 DBH (0.37) HTTSMN1; SMN2IDO1LMNAALDH1A1
SCHEMBL27731268 0.79 ICMT (0.52) MAPTLMNATP53RXFP1ICMT
SCHEMBL694560 0.77 TNF (0.44) KDM4ESMN1; SMN2LMNAALDH1A1TSHR
SCHEMBL3849945 0.75 ALDH1A1 (0.46) KDM4EHTTSMN1; SMN2MAPTLMNA
SCHEMBL27751731 0.74 KIF11 (0.42) MAPTLMNAICMTHTR6PTGS2
SCHEMBL3856954 0.74 AGXT (0.43) MAPTLMNAICMTHTR6PTGS2
SCHEMBL17956236 0.73 CNR1 (0.40) KDM4EMAPTALDH1A1HTR6
SCHEMBL27905750 0.73 HTT (0.49) HTTSMN1; SMN2IDO1MAPTLMNA
SCHEMBL6087143 0.73 HTR6 (0.54) KDM4EHTTSMN1; SMN2HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1956910-A2 ONCOGENIC RAS-SPECIFIC CYTOTOXIC COMPOUND AND METHODS OF USE THEREOF The Board of Regents of The University of Texas System (US) 2008-08-20 EP disclosed
WO-2007062399-A2 ONCOGENIC RAS-SPECIFIC CYTOTOXIC COMPOUND AND METHODS OF USE THEREOF THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2007-05-31 WO disclosed