SCHEMBL5144476

SCHEMBL5144476

COc1[nH]c2ccccc2c1CC#N

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 5/20 0.58
SRC P12931 2/20 0.58
KDM4E B2RXH2 6/20 0.45
FNTA P49354 1/20 0.41
FNTB P49356 1/20 0.41
MAPT P10636 4/20 0.40
ATM Q13315 1/20 0.40
ALDH1A1 P00352 5/20 0.39
HSD17B10 Q99714 2/20 0.39
CYP3A4 P08684 1/20 0.39
MEN1 O00255 1/20 0.39
HPGD P15428 1/20 0.39
KMT2A Q03164 1/20 0.39
MGAM O43451 1/20 0.39
TSHR P16473 1/20 0.38
HTT P42858 1/20 0.38
TUBB4A P04350 2/20 0.38
TUBB P07437 2/20 0.38
TUBA3C P0DPH7 2/20 0.38
TUBA1B P68363 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5767867 0.79 EGFR (0.52) EGFRSRCKDM4EFNTAFNTB
SCHEMBL28012374 0.78 ALDH1A1 (0.49) EGFRSRCKDM4EMAPTATM
SCHEMBL7127234 0.78 EGFR (0.63) EGFRSRCKDM4EMAPTALDH1A1
SCHEMBL29915686 0.78 EGFR (0.63) EGFRSRCKDM4EMAPTALDH1A1
SCHEMBL3868019 0.75 MAPT (0.65) EGFRKDM4EMAPTATMALDH1A1
SCHEMBL29128851 0.75 HTR6 (0.52) EGFRSRCKDM4EMAPTATM
SCHEMBL3221608 0.75 EGFR (0.59) EGFRSRCKDM4EFNTAFNTB
SCHEMBL9503673 0.75 KDM4E (0.52) EGFRSRCKDM4EMAPTALDH1A1
SCHEMBL6669729 0.75 EGFR (0.63) EGFRSRCKDM4EFNTAFNTB
SCHEMBL5571976 0.75 KDM4E (0.48) KDM4EMAPTATMALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1499188-A4 TOBACCO HAVING REDUCED NICOTINE AND NITROSAMINES VECTOR TOBACCO LTD (BM) 2007-11-14 EP disclosed
EP-1499188-A1 TOBACCO HAVING REDUCED NICOTINE AND NITROSAMINES Vector Tobacco Ltd. (BM) 2005-01-26 EP disclosed
WO-2003086076-A1 TOBACCO HAVING REDUCED NICOTINE AND NITROSAMINES VECTOR TOBACCO LTD. (BM) 2003-10-23 WO disclosed