SCHEMBL5147203

SCHEMBL5147203

CCN(CC1CCC1)c1ccc2c(c1C(C)N(Cc1cc(C#N)cc(C(F)(F)F)c1)C(=O)O)CCCC2

nearest known ligand 0.33

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 1/20 0.33
RXRA P19793 1/20 0.33
RXRG P48443 1/20 0.33
CETP P11597 2/20 0.32
PDE2A O00408 1/20 0.31
PTGES O14684 1/20 0.30
EP300 Q09472 1/20 0.30
CREBBP Q92793 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5149805 0.99 CCR2 (0.33) CCR2RXRARXRGCETPPDE2A
SCHEMBL5148371 0.98 CCR2 (0.33) CCR2RXRARXRGCETPPDE2A
SCHEMBL5150957 0.91 CCR2 (0.33) CCR2RXRARXRGCETPPDE2A
SCHEMBL1897361 0.85 CETP (0.33) CCR2RXRARXRGCETPPTGES
SCHEMBL5670667 0.84 RXRA (0.34) CCR2RXRARXRGCETPPDE2A
SCHEMBL5148310 0.83 RXRA (0.34) CCR2RXRARXRGCETPPDE2A
SCHEMBL5670023 0.82 RXRA (0.34) CCR2RXRARXRGCETPPDE2A
SCHEMBL1897741 0.80 CETP (0.41) CCR2CETP
SCHEMBL1897159 0.78 CETP (0.41) CETP
SCHEMBL5670569 0.78 CCR2 (0.31) CCR2RXRARXRG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070054839-A1 Method of inhibiting remnant lipoprotein production JAPAN TOBACCO INC. (JP) 2007-03-08 US claimed
US-20060270705-A1 Method for inhibiting lipid absorption and lipid absorption inhibitor JAPAN TOBACCO INC. (JP) 2006-11-30 US claimed
US-20070054839-A1 Method of inhibiting remnant lipoprotein production JAPAN TOBACCO INC. (JP) 2007-03-08 US disclosed
US-20060270705-A1 Method for inhibiting lipid absorption and lipid absorption inhibitor JAPAN TOBACCO INC. (JP) 2006-11-30 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070054839-A1 Method of inhibiting remnant lipoprotein production CETP, PCSK9, LIPA CCR2 2812/4885RXRA 2112/4885RXRG 2127/4885
US-20060270705-A1 Method for inhibiting lipid absorption and lipid absorption inhibitor CETP, SI, LIPC CCR2 4155/4885RXRA 3574/4885RXRG 3256/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.