SCHEMBL5147376

SCHEMBL5147376

CC(C)(OC(=O)c1ccccc1)OC(=O)C(N)C1(CC(=O)O)CCCCC1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 4/20 0.36
CYP1A2 P05177 3/20 0.36
CYP2C19 P33261 2/20 0.36
SLC6A3 Q01959 2/20 0.36
SLC6A2 P23975 1/20 0.36
SLC6A4 P31645 1/20 0.36
ADRB2 P07550 2/20 0.36
ADRB1 P08588 2/20 0.36
ADRB3 P13945 2/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
SLC7A5 Q01650 1/20 0.36
MAPK1 P28482 2/20 0.35
HIF1A Q16665 1/20 0.35
TSHR P16473 3/20 0.34
ALDH1A1 P00352 2/20 0.34
LMNA P02545 2/20 0.34
TDP1 Q9NUW8 2/20 0.34
HSD17B10 Q99714 1/20 0.34
SCN1A P35498 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3817343 0.82 USP2 (0.36) CYP1A2CYP2C19TSHRALDH1A1LMNA
SCHEMBL25013 0.81 LMNA (0.41) CYP2D6CYP1A2CYP2C19SLC6A3SLC6A2
SCHEMBL5148738 0.81 USP2 (0.35) CYP1A2CYP2C19TSHRALDH1A1LMNA
SCHEMBL4756226 0.80 USP2 (0.34) CYP1A2CYP2C19TSHRALDH1A1LMNA
SCHEMBL27641457 0.80 ADRB2 (0.43) CYP2D6CYP1A2SLC6A3SLC6A2SLC6A4
SCHEMBL4756846 0.79 USP2 (0.33) CYP1A2CYP2C19TSHRALDH1A1LMNA
SCHEMBL1076766 0.78 USP2 (0.39) CYP1A2CYP2C19TSHRALDH1A1LMNA
SCHEMBL4756232 0.78 TP53 (0.38) CYP2D6CYP1A2CYP2C19SLC6A3SLC6A2
SCHEMBL4756193 0.78 LMNA (0.36) CYP2D6CYP1A2CYP2C19SLC6A3SLC6A2
SCHEMBL6884986 0.77 TP53 (0.37) CYP2D6CYP1A2SLC6A3SLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1569895-A4 PRODRUGS OF GABA ANALOGS, COMPOSITIONS AND USES THEREOF XENOPORT INC (US) 2007-07-11 EP disclosed
EP-1569895-A1 PRODRUGS OF GABA ANALOGS, COMPOSITIONS AND USES THEREOF Xenoport, Inc. (US) 2005-09-07 EP disclosed
WO-2004052844-A1 PRODRUGS OF GABA ANALOGS, COMPOSITIONS AND USES THEREOF XENOPORT, INC. (US) 2004-06-24 WO disclosed