SCHEMBL5148906

SCHEMBL5148906

COc1ccc2c(C)c(S(=O)(=O)Cl)sc2c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.47
NPSR1 Q6W5P4 2/20 0.47
PRNP P04156 1/20 0.47
TSHR P16473 1/20 0.47
MAPK1 P28482 1/20 0.47
PPARG P37231 1/20 0.47
HTT P42858 1/20 0.47
MAPK10 P53779 1/20 0.47
NCOA2 Q15596 1/20 0.47
RXFP1 Q9HBX9 1/20 0.47
ALDH1A1 P00352 6/20 0.44
MAPT P10636 6/20 0.44
KDM4E B2RXH2 4/20 0.44
GAA P10253 2/20 0.44
LMNA P02545 2/20 0.44
CA2 P00918 2/20 0.42
KMT2A Q03164 3/20 0.41
HSD17B10 Q99714 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL787547 0.88 L3MBTL1 (0.50) NPSR1TSHRALDH1A1MAPTKDM4E
SCHEMBL14620656 0.86 CES2 (0.48) CES2NPSR1PRNPTSHRMAPK1
SCHEMBL788639 0.80 NPSR1 (0.48) NPSR1RXFP1MAPTKMT2ANPC1
SCHEMBL14409807 0.75 CES2 (0.51) CES2NPSR1PRNPTSHRMAPK1
SCHEMBL14620655 0.74 L3MBTL1 (0.48) NPSR1TSHRALDH1A1MAPTKDM4E
SCHEMBL787663 0.74 HSD11B1 (0.43) NPSR1PRNPRXFP1ALDH1A1MAPT
SCHEMBL30017661 0.73 KDM4E (0.67) CES2NPSR1PRNPTSHRMAPK1
SCHEMBL13338880 0.73 KDM4E (0.67) CES2NPSR1PRNPTSHRMAPK1
SCHEMBL10369463 0.73 CA2 (0.52) CES2NPSR1PRNPTSHRMAPK1
SCHEMBL806148 0.73 L3MBTL1 (0.47) NPSR1ALDH1A1MAPTKDM4ECA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7157454-B2 Derivatives of n-(arylsulfonyl)beta-aminoacids comprising a substituted aminomethyl group, the preparation method thereof and the pharmaceutical compositions containing same SANOFI-AVENTIS (FR) 2007-01-02 US disclosed
US-20040116353-A1 Derivatives of n-(arylsulfonyl)beta-aminoacids comprising a substituted aminomethyl group, the preparation method thereof and the pharmaceutical compositions containing same SANOFI (FR) 2004-06-17 US disclosed