SCHEMBL5153249

SCHEMBL5153249

CCCN(C)C(=O)c1cc(C(=O)O)cc(-c2nccs2)c1.COC(=O)c1cc(I)cc(C(=O)O)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 1/20 0.36
SMPD3 Q9NY59 1/20 0.34
HPGD P15428 3/20 0.34
SLC6A9 P48067 1/20 0.33
HDAC2 Q92769 1/20 0.32
KDM4E B2RXH2 2/20 0.32
KDM6B O15054 1/20 0.32
KDM5C P41229 1/20 0.32
KDM4C Q9H3R0 1/20 0.32
KDM2A Q9Y2K7 1/20 0.32
KDM3A Q9Y4C1 1/20 0.32
ABL1 P00519 1/20 0.32
BCR P11274 1/20 0.32
ALDH1A1 P00352 3/20 0.31
PPARG P37231 1/20 0.31
MAPK10 P53779 1/20 0.31
KMT2A Q03164 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
RXFP1 Q9HBX9 1/20 0.31
NCOR2 Q9Y618 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3351720 0.91 SMPD3 (0.40) LTA4HSMPD3HPGDSLC6A9KDM4E
SCHEMBL3860707 0.88 LTA4H (0.38) LTA4HSMPD3HPGDSLC6A9HDAC2
SCHEMBL13306591 0.85 ALDH1A1 (0.43) LTA4HSMPD3HPGDSLC6A9KDM4E
SCHEMBL3347738 0.82 SMPD3 (0.41) LTA4HSMPD3HPGDSLC6A9KDM4E
SCHEMBL3350524 0.82 LTA4H (0.39) LTA4HSMPD3HPGDSLC6A9ABL1
SCHEMBL3355550 0.80 LMNA (0.42) KDM4EALDH1A1KMT2AMAPTTDP1
SCHEMBL3348439 0.78 F2 (0.39) LTA4HSMPD3HPGDSLC6A9HDAC2
SCHEMBL3860120 0.77 TPMT (0.40) KDM4EALDH1A1KMT2A
SCHEMBL3350413 0.73 ESR1 (0.41) HPGDKDM4EALDH1A1MAPTTDP1
SCHEMBL5155253 0.73 PLA2G2A (0.47) KDM4EKDM6BKDM5CKDM4CKDM2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1740573-A1 AMIDES AS BACE INHIBITORS ELI LILLY AND COMPANY (US) 2007-01-10 EP disclosed
EP-1740575-A2 PYRROLIDINE DERIVATIVES USEFUL AS BACE INHIBITORS ELI LILLY AND COMPANY (US) 2007-01-10 EP disclosed
WO-2005108358-A2 PYRROLIDINE DERIVATIVES USEFUL AS BACE INHIBITORS ELI LILLY AND COMPANY (US) 2005-11-17 WO disclosed
WO-2005108391-A1 AMIDES AS BACE INHIBITORS ELI LILLY AND COMPANY (US) 2005-11-17 WO disclosed