SCHEMBL5158048

SCHEMBL5158048

CCC(C)c1ccc(NC(=O)CCC(=O)NC2CCC(Cc3ccc(Cl)cc3)(N(C)C)CC2)cc1.O=C(O)CCCC(=O)N1CC=C(c2ccccc2)CC1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 10/20 0.38
CNR1 P21554 1/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
ALDH1A1 P00352 2/20 0.37
TP53 P04637 1/20 0.37
MAPT P10636 1/20 0.37
ALOX12 P18054 1/20 0.37
HTT P42858 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
CCR1 P32246 1/20 0.34
DGAT1 O75907 1/20 0.34
POLB P06746 1/20 0.33
PSMB11 A5LHX3 1/20 0.33
PSMA7 O14818 1/20 0.33
PSMB1 P20618 1/20 0.33
PSMA1 P25786 1/20 0.33
PSMA2 P25787 1/20 0.33
PSMA3 P25788 1/20 0.33
PSMA4 P25789 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL207100 0.83 NPSR1 (0.43) MEN1KMT2AALDH1A1TP53MAPT
SCHEMBL206590 0.81 MEN1 (0.47) NAMPTMEN1KMT2AALDH1A1TP53
SCHEMBL205784 0.79 MEN1 (0.49) NAMPTMEN1KMT2AALDH1A1TP53
SCHEMBL205169 0.78 SIGMAR1 (0.41) CNR1MEN1KMT2AALDH1A1MAPT
SCHEMBL207488 0.74 MEN1 (0.47) MEN1KMT2AALDH1A1TP53MAPT
SCHEMBL5158010 0.74 OPRM1 (0.40) CNR1MEN1KMT2AALDH1A1TP53
SCHEMBL5158031 0.73 KMT2A (0.52) NAMPTMEN1KMT2AALDH1A1TP53
SCHEMBL5160624 0.71 LMNA (0.43) MEN1KMT2AALDH1A1TP53SMN1; SMN2
SCHEMBL205873 0.70 UTS2R (0.43) KMT2APOLB
SCHEMBL205853 0.70 HPGD (0.40) MEN1KMT2AALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1745010-A1 SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES Grünenthal GmbH (DE) 2007-01-24 EP disclosed
WO-2005110974-A1 SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES Grünenthal GmbH (DE) 2005-11-24 WO disclosed