SCHEMBL5158160

SCHEMBL5158160

CCNC(=O)CC(=O)c1cn[nH]c1

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ACACB O00763 3/20 0.37
ROCK2 O75116 2/20 0.36
ROCK1 Q13464 2/20 0.36
NAMPT P43490 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.35
NOS2 P35228 1/20 0.34
BAZ2B Q9UIF8 1/20 0.34
BAZ2A Q9UIF9 1/20 0.34
ALDH1A1 P00352 1/20 0.34
HTT P42858 1/20 0.34
KDM4E B2RXH2 1/20 0.33
MAPK1 P28482 1/20 0.33
HPGD P15428 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5161535 0.83 ALDH1A1 (0.39) ACACBROCK2ROCK1NOS2BAZ2B
SCHEMBL1608977 0.82 ROCK2 (0.47) ACACBROCK2ROCK1NAMPT
SCHEMBL8402539 0.78
SCHEMBL5160875 0.77 MEN1 (0.41) ACACBROCK2ROCK1NAMPTNOS2
SCHEMBL20797184 0.77 ALDH1A1 (0.38) ACACBROCK2ROCK1NOS2ALDH1A1
SCHEMBL5162787 0.77 KMT2A (0.53) ACACBNAMPTALDH1A1KDM4EHPGD
SCHEMBL5163272 0.75 ACACB (0.39) ACACBROCK2NAMPTNOS2ALDH1A1
SCHEMBL5178020 0.75 NOS2 (0.38) ACACBROCK1NOS2ALDH1A1HTT
SCHEMBL20992124 0.75 HSD17B3 (0.46) ACACBL3MBTL1NOS2ALDH1A1HTT
SCHEMBL5163553 0.75 ACACB (0.38) ACACBROCK2NAMPTNOS2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8293899-B2 Ketone transfer hydrogenation of stereoisomerically enriched 3-heteroaryl-3-oxocarboxylic esters by reducing 3-heteroaryl-3-hydroxycarboxylic esters in the presence of a ruthenium-containing catalyst, an amine and formic acid and/or formates LANXESS DEUTSCHLAND GMBH (DE) 2012-10-23 US disclosed
EP-1340746-B1 Process for the reduction of 3-heteroaryl-3-oxo-propanoic acid derivatives SALTIGO GMBH (DE) 2007-02-28 EP disclosed
US-20030225274-A1 Process for reducing 3-heteroaryl-3-oxopropionic acid derivatives LANXESS DEUTSCHLAND GMBH (DE) 2003-12-04 US disclosed
EP-1340746-A1 Process for the reduction of 3-heteroaryl-3-oxo-propanoic acid derivatives BAYER AG (DE) 2003-09-03 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030225274-A1 Process for reducing 3-heteroaryl-3-oxopropionic acid derivatives GRHPR, HPD, HAAO ACACB 76/4885ROCK2 4242/4885ROCK1 4411/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.