SCHEMBL5158447

SCHEMBL5158447

COc1c(N2CCOC2=O)cc(N2CCOC2=O)c(C)c1C

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.36
CRHR1 P34998 1/20 0.35
PIK3CA P42336 1/20 0.34
MTOR P42345 1/20 0.34
MAPK10 P53779 1/20 0.33
MET P08581 1/20 0.33
NPSR1 Q6W5P4 1/20 0.32
IDH1 O75874 1/20 0.32
RXFP1 Q9HBX9 1/20 0.32
PKM P14618 1/20 0.32
TYK2 P29597 1/20 0.32
TSHR P16473 1/20 0.31
NQO2 P16083 1/20 0.31
PDE10A Q9Y233 1/20 0.31
PARP1 P09874 1/20 0.31
DPP4 P27487 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5176620 0.95 ALDH1A1 (0.37) ALDH1A1CRHR1PIK3CAMTORMAPK10
SCHEMBL5692224 0.86 PIK3CA (0.37) ALDH1A1CRHR1PIK3CAMTORMAPK10
SCHEMBL5486206 0.81 ALDH1A1 (0.37) ALDH1A1CRHR1PIK3CAMTORMAPK10
SCHEMBL5691400 0.78 P2RX7 (0.39) ALDH1A1PIK3CAMTORMAPK10MET
Hydrochloric Acid SCHEMBL9461657 0.76 HTR1A (0.34) ALDH1A1CRHR1PIK3CAMTORMAPK10
SCHEMBL30602382 0.76 P2RX7 (0.38) CRHR1PIK3CAMTORMAPK10MET
SCHEMBL29130967 0.76 P2RX7 (0.38) CRHR1PIK3CAMTORMAPK10MET
SCHEMBL5175915 0.73 CMA1 (0.35) PIK3CAMTORIDH1PARP1
SCHEMBL6264641 0.73 SYK (0.36) ALDH1A1CRHR1PIK3CAMTORMAPK10
SCHEMBL9461697 0.72 GRIN2D (0.43) ALDH1A1PKMTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1748822-A1 M-PHENYLENE DIAMINE COUPLING COMPONENTS Henkel Kommanditgesellschaft auf Aktien (DE) 2007-02-07 EP claimed
WO-2005117819-A1 M-PHENYLENE DIAMINE COUPLING COMPONENTS HENKEL KOMMANDITGESELLSCHAFT AUF AKTIEN (DE) 2005-12-15 WO claimed
EP-1748822-A1 M-PHENYLENE DIAMINE COUPLING COMPONENTS Henkel Kommanditgesellschaft auf Aktien (DE) 2007-02-07 EP disclosed
WO-2005117819-A1 M-PHENYLENE DIAMINE COUPLING COMPONENTS HENKEL KOMMANDITGESELLSCHAFT AUF AKTIEN (DE) 2005-12-15 WO disclosed