SCHEMBL5159963

SCHEMBL5159963

O=C(NO)O[C@@H]1c2ccccc2CCN1S(=O)(=O)c1ccc(Oc2ccc(F)cc2)cc1

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.49
MMP3 P08254 9/20 0.49
MMP9 P14780 4/20 0.49
MMP2 P08253 3/20 0.49
MMP1 P03956 10/20 0.49
MMP7 P09237 5/20 0.48
ADAM17 P78536 3/20 0.47
MMP8 P22894 6/20 0.47
SMN1; SMN2 Q16637 1/20 0.46
MMP13 P45452 2/20 0.45
MMP12 P39900 1/20 0.42
MMP14 P50281 1/20 0.42
MMP15 P51511 1/20 0.42
MMP16 P51512 1/20 0.42
MMP26 Q9NRE1 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5160245 1.00 THRB (0.49) THRBMMP3MMP9MMP2MMP1
SCHEMBL5164049 0.90 MMP1 (0.52) MMP3MMP9MMP2MMP1MMP7
SCHEMBL5160366 0.90 MMP1 (0.51) MMP3MMP9MMP2MMP1MMP7
SCHEMBL5160300 0.89 MMP8 (0.49) MMP3MMP9MMP2MMP1MMP7
SCHEMBL4693205 0.89 MMP1 (0.47) MMP3MMP9MMP2MMP1MMP7
SCHEMBL5162513 0.89 MMP1 (0.47) MMP3MMP9MMP2MMP1MMP7
SCHEMBL5163119 0.89 MMP1 (0.47) MMP3MMP9MMP2MMP1MMP7
SCHEMBL5165012 0.89 MMP1 (0.48) MMP3MMP9MMP2MMP1MMP7
SCHEMBL5160395 0.89 MMP8 (0.60) THRBMMP3MMP9MMP2MMP1
SCHEMBL5443161 0.88 THRB (0.49) THRBMMP3MMP9MMP2MMP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1763516-A2 SUBSTITUTED TETRAHYDROISOCHINOLINES USED IN THE FORM OF MMP INHIBITORS, METHOD FOR THE PRODUCTION AND USE THEREOF IN THE FORM OF DRAGS Sanofi-Aventis Deutschland GmbH (DE) 2007-03-21 EP disclosed
WO-2006002763-A2 SUBSTITUTED TETRAHYDROISOCHINOLINES USED IN THE FORM OF MMP INHIBITORS, METHOD FOR THE PRODUCTION AND USE THEREOF IN THE FORM OF DRAGS SANOFI-AVENTIS DEUTSCHLAND GMBH (DE) 2006-01-12 WO disclosed