SCHEMBL5162823

SCHEMBL5162823

CC(C)(C)OC(=O)ON1CCC(N2CCC(C#N)CC2)CC1

nearest known ligand 0.35

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM2B Q8NHM5 1/20 0.35
CTSK P43235 3/20 0.34
AOC3 Q16853 1/20 0.32
CHRM1 P11229 2/20 0.32
IRAK4 Q9NWZ3 1/20 0.32
MEN1 O00255 1/20 0.32
ALDH1A1 P00352 1/20 0.32
MAPT P10636 1/20 0.32
KMT2A Q03164 1/20 0.32
OPRM1 P35372 2/20 0.31
OPRD1 P41143 2/20 0.31
OGFRL1 Q5TC84 2/20 0.31
DPP4 P27487 1/20 0.31
HPGD P15428 1/20 0.31
GPR119 Q8TDV5 1/20 0.31
CHRM2 P08172 1/20 0.31
CHRM3 P20309 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2087178 0.82 HPGD (0.48) CHRM1MEN1ALDH1A1MAPTKMT2A
SCHEMBL16341947 0.82 CHRM1 (0.34) CHRM1OPRM1OPRD1OGFRL1HPGD
SCHEMBL4046200 0.79 L3MBTL3 (0.33) CHRM1KMT2AHPGDCHRM2CHRM3
SCHEMBL27997009 0.78 CTSK (0.35) CTSKMEN1ALDH1A1MAPTKMT2A
SCHEMBL4046093 0.77 HRH3 (0.35) CTSKCHRM1MEN1ALDH1A1MAPT
SCHEMBL31209769 0.76 MAPT (0.47) MEN1ALDH1A1MAPTKMT2ADPP4
SCHEMBL4716959 0.75 DRD2 (0.38) CHRM1CHRM2CHRM3
SCHEMBL4593426 0.74 KMT2A (0.34) MEN1ALDH1A1MAPTKMT2AOPRM1
SCHEMBL4067285 0.74 CHRM2 (0.36) CTSKCHRM1GPR119CHRM2CHRM3
SCHEMBL4658596 0.74 CHRM2 (0.33) CHRM1IRAK4MEN1KMT2AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1770086-A1 Selected CGRP antagonists, process for their preparation as well as their use as medicaments Boehringer Ingelheim Pharma GmbH & Co. KG (DE) 2007-04-04 EP disclosed