SCHEMBL5163365

SCHEMBL5163365

Cc1c(-c2ccc(C[C@@H](C(=O)O)N(C(=O)OC(C)(C)C)C(=O)[C@@H]3CCCN3)cc2)c(=O)n(C)c(=O)n1C

nearest known ligand 0.42

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 14/20 0.42
ITGB7 P26010 14/20 0.42
ITGB1 P05556 12/20 0.42
SCN9A Q15858 1/20 0.32
SCN3A Q9NY46 1/20 0.32
SCN5A Q14524 1/20 0.32
CTSC P53634 3/20 0.31
CTSK P43235 1/20 0.31
SCN4A P35499 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5162837 0.93 ITGA4 (0.42) ITGA4ITGB7ITGB1SCN9ASCN3A
SCHEMBL3165698 0.81 CTSC (0.43) CTSCSCN4A
SCHEMBL5162144 0.76 ITGB1 (0.58) ITGA4ITGB7ITGB1CTSCCTSK
Hydrochloric Acid SCHEMBL5160248 0.75 ITGB1 (0.57) ITGA4ITGB7ITGB1CTSCCTSK
Hydrochloric Acid SCHEMBL7423666 0.75 ITGB1 (0.57) ITGA4ITGB7ITGB1CTSCCTSK
SCHEMBL5163361 0.68 ITGA4 (0.55) ITGA4ITGB7ITGB1
SCHEMBL27514790 0.68 ITGB3 (0.33) SCN4A
SCHEMBL3656054 0.67 CTSC (0.47) CTSCCTSK
SCHEMBL6368640 0.67 HTR2C (0.43) CTSCSCN4A
SCHEMBL27735771 0.67 ITGB3 (0.45) ITGA4ITGB7CTSC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1237878-B1 4-PYRIMIDINYL-N-ACYL-L-PHENYLALANINES HOFFMANN LA ROCHE (CH) 2007-03-21 EP disclosed
EP-1237878-A2 4-PYRIMIDINYL-N-ACYL-L-PHENYLALANINES F. HOFFMANN-LA ROCHE AG (CH) 2002-09-11 EP disclosed
US-6380387-B1 ANTIINFLAMMATORY AGENTS, ANTIASTHMATICS HOFFMANN-LA ROCHE INC. 2002-04-30 US disclosed
WO-2001042225-A2 4-PYRIMIDINYL-N-ACYL-L-PHENYLALANINES F. HOFFMANN-LA ROCHE AG (CH) 2001-06-14 WO disclosed