SCHEMBL5164161

SCHEMBL5164161

O=C(O)OC1CCCN1C(=O)Nc1ccccc1

nearest known ligand 0.62

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.62
NPC1 O15118 3/20 0.62
RAB9A P51151 2/20 0.62
POLB P06746 1/20 0.54
CYP2C9 P11712 1/20 0.54
CYP2C19 P33261 1/20 0.54
ALDH1A1 P00352 4/20 0.51
FKBP1A P62942 2/20 0.51
THRB P10828 1/20 0.49
ALOX12 P18054 1/20 0.49
KMT2A Q03164 1/20 0.49
MAPT P10636 1/20 0.49
TP53 P04637 1/20 0.48
HTT P42858 2/20 0.47
BCHE P06276 2/20 0.46
MAOB P27338 1/20 0.46
KDM4E B2RXH2 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5161696 0.88 SMN1; SMN2 (0.53) SMN1; SMN2NPC1RAB9ACYP2C9CYP2C19
SCHEMBL31234028 0.78 SMN1; SMN2 (0.67) SMN1; SMN2NPC1RAB9APOLBCYP2C9
SCHEMBL4186674 0.78 KMT2A (0.76) SMN1; SMN2NPC1RAB9APOLBCYP2C9
SCHEMBL27627515 0.77 ALDH1A1 (0.79) SMN1; SMN2NPC1RAB9ACYP2C9CYP2C19
SCHEMBL5734401 0.75 NPC1 (0.63) SMN1; SMN2NPC1RAB9APOLBCYP2C9
SCHEMBL11719448 0.75 KMT2A (0.70) SMN1; SMN2NPC1RAB9APOLBCYP2C9
Iodide SCHEMBL10827466 0.74 NPC1 (0.62) SMN1; SMN2NPC1RAB9APOLBCYP2C9
SCHEMBL11181068 0.74 SMN1; SMN2 (0.62) SMN1; SMN2NPC1RAB9APOLBCYP2C9
SCHEMBL7309663 0.74 THRB (0.70) SMN1; SMN2NPC1RAB9APOLBCYP2C9
SCHEMBL3433977 0.74 SMN1; SMN2 (0.65) SMN1; SMN2NPC1RAB9APOLBCYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2051975-B1 SUBSTITUTED PROLINAMIDES, PRODUCTION THEREOF AND THEIR USE AS DRUGS BOEHRINGER INGELHEIM INT (DE) 2012-09-12 EP disclosed
EP-1760081-A1 Method for the production of pyrrolidine-1,2-dicarboxylic acid-1-(phenyl(-amide))-2-(phenyl(-amide)) derivatives and 1-(phenylcarbamoyl)-pyrrolidine-2-carboxylic acid derivatives as intermediate products Merck Patent GmbH (DE) 2007-03-07 EP disclosed