SCHEMBL5165883

SCHEMBL5165883

Nc1cc2c(cc1OCc1cccnc1)OCCO2

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.45
DRD2 P14416 2/20 0.45
SMN1; SMN2 Q16637 1/20 0.44
CYP11B1 P15538 2/20 0.43
CYP11B2 P19099 2/20 0.43
CYP19A1 P11511 1/20 0.43
CLK4 Q9HAZ1 1/20 0.43
IKBKB O14920 1/20 0.43
VNN1 O95497 1/20 0.42
SLC6A4 P31645 1/20 0.42
MAOA P21397 1/20 0.42
MAOB P27338 1/20 0.42
OGA O60502 1/20 0.41
MAP4K3 Q8IVH8 1/20 0.40
CHEK1 O14757 1/20 0.40
HTR6 P50406 1/20 0.40
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
GAA P10253 1/20 0.40
MAPT P10636 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17323482 0.83 HTR1A (0.54) HTR1ADRD2CYP11B1CYP11B2CYP19A1
SCHEMBL21213375 0.78 MAOB (0.69) SMN1; SMN2CYP11B1CYP11B2VNN1MAOA
Hydrochloric Acid SCHEMBL5166479 0.78 CYP11B1 (0.45) HTR1ADRD2SMN1; SMN2CYP11B1CYP11B2
SCHEMBL13428030 0.76 CYP19A1 (0.58) HTR1ADRD2CYP11B1CYP11B2CYP19A1
SCHEMBL1028598 0.74 HTR1A (0.61) HTR1ADRD2CYP11B1CYP11B2CYP19A1
SCHEMBL2038362 0.74 HTR1A (0.51) HTR1ADRD2CYP11B1CYP11B2CYP19A1
SCHEMBL3315005 0.74 HTR1A (0.51) HTR1ADRD2CYP11B1CYP11B2CYP19A1
SCHEMBL2038082 0.74 LRRK2 (0.50) HTR1ADRD2CYP11B1CYP11B2CYP19A1
SCHEMBL5165973 0.73 LMNA (0.42) HTR1ADRD2CYP11B1CYP11B2CYP19A1
SCHEMBL29857565 0.71 LTA4H (0.73) HTR1ADRD2SMN1; SMN2CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1765808-A1 BISARYLUREA DERIVATIVES USEFUL FOR INHIBITING CHK1 ICOS Corporation (US) 2007-03-28 EP disclosed
WO-2006012308-A1 BISARYLUREA DERIVATIVES USEFUL FOR INHIBITING CHK1 ICOS CORPORATION (US) 2006-02-02 WO disclosed