SCHEMBL5169062

SCHEMBL5169062

COc1ccc(CC(=O)NOCCc2ccccc2)cc1

nearest known ligand 0.62

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.62
NPC1 O15118 2/20 0.62
RAB9A P51151 3/20 0.59
MAPT P10636 2/20 0.59
SMN1; SMN2 Q16637 1/20 0.59
CNR2 P34972 1/20 0.57
HTT P42858 1/20 0.56
PLAU P00749 1/20 0.56
ELANE P08246 1/20 0.56
EGFR P00533 1/20 0.54
ERBB2 P04626 1/20 0.54
ALOX5 P09917 1/20 0.54
MEN1 O00255 1/20 0.52
KMT2A Q03164 1/20 0.52
ATM Q13315 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4917828 0.86 RAB9A (0.68) ALDH1A1NPC1RAB9AMAPTSMN1; SMN2
SCHEMBL8691052 0.80 MAPT (0.76) ALDH1A1NPC1RAB9AMAPT
SCHEMBL22283905 0.79 SMN1; SMN2 (0.61) ALDH1A1NPC1RAB9AMAPTSMN1; SMN2
SCHEMBL4928502 0.77 HTT (0.73) ALDH1A1NPC1RAB9AMAPTSMN1; SMN2
SCHEMBL28497417 0.77 NPC1 (1.00) ALDH1A1NPC1RAB9AMAPTSMN1; SMN2
SCHEMBL5862101 0.77 NPC1 (1.00) ALDH1A1NPC1RAB9AMAPTSMN1; SMN2
SCHEMBL8938110 0.76 HDAC8 (0.53) ALDH1A1RAB9AMAPTSMN1; SMN2CNR2
SCHEMBL4032340 0.75 NPC1 (0.66) ALDH1A1NPC1RAB9AMAPTSMN1; SMN2
SCHEMBL6938387 0.75 NPC1 (0.55) ALDH1A1NPC1RAB9AMAPTSMN1; SMN2
SCHEMBL6171613 0.75 RAB9A (1.00) ALDH1A1NPC1RAB9AMAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1771410-A1 SPIROLACTAMS AND THEIR SYNTHESIS LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2007-04-11 EP disclosed
WO-2005108356-A1 SPIROLACTAMS AND THEIR SYNTHESIS LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2005-11-17 WO disclosed