Aziridine

Aziridine

SCHEMBL5185484

C1CN1.Cc1ccc(S(=O)(=O)O)cc1

nearest known ligand 0.50

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABL1BMXBRAFBTKCHRNA4CHRNB2CSNK1EEGFRERBB2F10FLT1FLT3FLT4IGF1RINSRITKJAK3KDRKITOPRM1PARP1PARP2PDGFRBPIK3CDRAF1RETSLC18A2TECTXKdacAdacBdacCftsImrcAmrcBmrdArplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Aziridine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.50
SMN1; SMN2 Q16637 3/20 0.50
LMNA P02545 2/20 0.50
HTT P42858 2/20 0.50
GAA P10253 2/20 0.50
MAPT P10636 2/20 0.50
KDM4E B2RXH2 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
CYP2D6 P10635 2/20 0.49
SNCA P37840 1/20 0.47
PKM P14618 3/20 0.47
CA1 P00915 2/20 0.47
CA2 P00918 2/20 0.47
MMP1 P03956 1/20 0.47
MMP2 P08253 1/20 0.47
MMP9 P14780 1/20 0.47
MMP8 P22894 1/20 0.47
MMP13 P45452 1/20 0.47
TSHR P16473 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Piperazine SCHEMBL5875357 0.98 ALDH1A1 (0.49) ALDH1A1SMN1; SMN2LMNAHTTGAA
Piperazine SCHEMBL7635861 0.98 ALDH1A1 (0.49) ALDH1A1SMN1; SMN2LMNAHTTGAA
Pyrrolidine SCHEMBL2531422 0.94 ALDH1A1 (0.46) ALDH1A1SMN1; SMN2LMNAHTTGAA
Azetidine SCHEMBL28290955 0.94 ALDH1A1 (0.49) ALDH1A1SMN1; SMN2LMNAHTTGAA
Piperidine SCHEMBL631560 0.92 ALDH1A1 (0.45) ALDH1A1SMN1; SMN2LMNAHTTGAA
Piperidine SCHEMBL4867261 0.92 ALDH1A1 (0.45) ALDH1A1SMN1; SMN2LMNAHTTGAA
Pyrrolidine SCHEMBL16241174 0.92 ALDH1A1 (0.45) ALDH1A1SMN1; SMN2LMNAHTTGAA
Piperidine SCHEMBL16927692 0.91 ALDH1A1 (0.44) ALDH1A1SMN1; SMN2LMNAHTTGAA
Morpholine SCHEMBL890524 0.89 L3MBTL1 (0.43) ALDH1A1SMN1; SMN2LMNAHTTGAA
SCHEMBL3739461 0.89 MAPT (0.44) ALDH1A1SMN1; SMN2LMNAHTTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1518908-B1 Ink composition for electrostatic ink-jet recording and method of ink-jet recording FUJIFILM CORP (JP) 2007-05-30 EP disclosed
US-20050070630-A1 Ink composition for electrostatic ink-jet recording and method of ink-jet recording FUJI PHOTO FILM CO., LTD. 2005-03-31 US disclosed
EP-1518908-A1 Ink composition for electrostatic ink-jet recording and method of ink-jet recording FUJI PHOTO FILM CO., LTD. (JP) 2005-03-30 EP disclosed