SCHEMBL5190965

SCHEMBL5190965

NC(=O)CC1CN(C(=O)c2cccnc2)CCN1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.51
CHRNB4 P30926 1/20 0.51
CHRNA3 P32297 1/20 0.51
CHRNA7 P36544 1/20 0.51
CHRNA4 P43681 1/20 0.51
GAA P10253 1/20 0.45
ALDH1A1 P00352 1/20 0.45
HPGD P15428 1/20 0.44
PKM P14618 1/20 0.44
MAPK1 P28482 1/20 0.44
CA1 P00915 4/20 0.44
CA2 P00918 4/20 0.44
CA4 P22748 4/20 0.44
CA9 Q16790 4/20 0.44
VNN1 O95497 1/20 0.44
POLB P06746 1/20 0.44
MKNK1 Q9BUB5 1/20 0.44
MKNK2 Q9HBH9 1/20 0.44
MEN1 O00255 1/20 0.43
MAPT P10636 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5193835 0.79 ALDH1A1 (0.48) CHRNB2CHRNB4CHRNA3CHRNA7CHRNA4
SCHEMBL5192050 0.77 CTSL (0.47) CHRNB2CHRNB4CHRNA3CHRNA7CHRNA4
SCHEMBL5192336 0.77 ALDH1A1 (0.51) GAAALDH1A1MEN1KMT2A
SCHEMBL5191569 0.77 ALDH1A1 (0.47) CHRNB2CHRNA4ALDH1A1MAPK1VNN1
SCHEMBL5206456 0.76 MAPK1 (0.58) ALDH1A1HPGDMAPK1POLBMEN1
SCHEMBL5206448 0.76 POLB (0.45) ALDH1A1MAPK1POLBMEN1KMT2A
SCHEMBL1088707 0.74 MKNK1 (0.72) CHRNB2CHRNB4CHRNA3CHRNA7CHRNA4
SCHEMBL29831536 0.74 MKNK1 (0.72) CHRNB2CHRNB4CHRNA3CHRNA7CHRNA4
SCHEMBL2628906 0.73 SIGMAR1 (0.59) CHRNB2CHRNB4CHRNA3CHRNA7CHRNA4
Hydrochloric Acid SCHEMBL9785721 0.73 MKNK1 (0.70) CHRNB2CHRNB4CHRNA3CHRNA7CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0968206-B8 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX INC (US) 2007-01-24 EP disclosed
EP-0968206-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 2000-01-05 EP disclosed
WO-1998037079-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 1998-08-27 WO disclosed