SCHEMBL5192050

SCHEMBL5192050

O=C(CC1CN(C(=O)c2cccnc2)CCN1)NCCc1cccs1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSL P07711 1/20 0.47
CTSB P07858 1/20 0.47
CASP3 P42574 1/20 0.47
CTSK P43235 1/20 0.47
CTSF Q9UBX1 1/20 0.47
CHRNB2 P17787 1/20 0.42
CHRNB4 P30926 1/20 0.42
CHRNA3 P32297 1/20 0.42
CHRNA7 P36544 1/20 0.42
CHRNA4 P43681 1/20 0.42
KMT2A Q03164 1/20 0.41
ROCK2 O75116 1/20 0.40
MC4R P32245 1/20 0.39
MC5R P33032 1/20 0.39
MC3R P41968 1/20 0.39
CHEK1 O14757 1/20 0.39
DAPK3 O43293 1/20 0.39
MAP4K4 O95819 1/20 0.39
PIM1 P11309 1/20 0.39
PRKACA P17612 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5281221 0.86 CTSL (0.51) CTSLCTSBCASP3CTSKCTSF
SCHEMBL5206456 0.80 MAPK1 (0.58) KMT2AALDH1A1MAPT
SCHEMBL5193835 0.78 ALDH1A1 (0.48) CHRNB2CHRNB4CHRNA3CHRNA7CHRNA4
SCHEMBL5190965 0.77 CHRNB2 (0.51) CHRNB2CHRNB4CHRNA3CHRNA7CHRNA4
SCHEMBL5191026 0.76 ADAM17 (0.43) KMT2AMC4RADAM17
SCHEMBL5192336 0.75 ALDH1A1 (0.51) KMT2AALDH1A1
SCHEMBL6320319 0.73 NOS2 (0.48) CTSLCTSBCASP3CTSKCTSF
SCHEMBL5192754 0.72 NOS2 (0.51) CTSLCTSBCASP3CTSKCTSF
SCHEMBL5193511 0.71 POLB (0.47) KMT2AMC4RADAM17
SCHEMBL5206448 0.69 POLB (0.45) CTSKKMT2AROCK2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0968206-B8 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX INC (US) 2007-01-24 EP claimed
EP-0968206-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 2000-01-05 EP claimed
WO-1998037079-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 1998-08-27 WO claimed