SCHEMBL5193835

SCHEMBL5193835

Cc1ccc(CNC(=O)CC2CN(C(=O)c3cccnc3)CCN2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.48
CHRNB2 P17787 1/20 0.44
CHRNB4 P30926 1/20 0.44
CHRNA3 P32297 1/20 0.44
CHRNA7 P36544 1/20 0.44
CHRNA4 P43681 1/20 0.44
NAMPT P43490 1/20 0.42
REN P00797 1/20 0.42
GAA P10253 1/20 0.42
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
FNTA P49354 1/20 0.41
FNTB P49356 1/20 0.41
MAPT P10636 1/20 0.40
HTT P42858 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
NOS2 P35228 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5192336 0.90 ALDH1A1 (0.51) ALDH1A1GAAMEN1KMT2A
SCHEMBL5206456 0.80 MAPK1 (0.58) ALDH1A1NAMPTMAPTHTTMEN1
SCHEMBL5190965 0.79 CHRNB2 (0.51) ALDH1A1CHRNB2CHRNB4CHRNA3CHRNA7
SCHEMBL5192050 0.78 CTSL (0.47) ALDH1A1CHRNB2CHRNB4CHRNA3CHRNA7
SCHEMBL5195331 0.73 GAA (0.49) ALDH1A1GAAMAPTHTTMEN1
SCHEMBL5206448 0.73 POLB (0.45) ALDH1A1HTTMEN1KMT2ASMN1; SMN2
SCHEMBL5193739 0.72 PKM (0.56) ALDH1A1MAPTMEN1KMT2ASMN1; SMN2
SCHEMBL5191591 0.72 TP53 (0.53) MAPTMEN1KMT2ASMN1; SMN2
SCHEMBL5193335 0.71 SMN1; SMN2 (0.49) ALDH1A1NAMPTGAACYP3A4CYP2C9
SCHEMBL5192010 0.71 HPGD (0.46) ALDH1A1MEN1KMT2ANOS2SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0968206-B8 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX INC (US) 2007-01-24 EP claimed
EP-0968206-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 2000-01-05 EP claimed
WO-1998037079-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 1998-08-27 WO claimed