SCHEMBL5192001

SCHEMBL5192001

CCCCN1CCN(Cc2ccc(C)cc2)C(CC(N)=O)C1

nearest known ligand 0.56

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 3/20 0.56
ALDH1A1 P00352 2/20 0.53
HTT P42858 2/20 0.52
PKM P14618 1/20 0.47
MEN1 O00255 4/20 0.47
KMT2A Q03164 4/20 0.47
POLB P06746 2/20 0.47
L3MBTL1 Q9Y468 1/20 0.45
GAA P10253 1/20 0.42
MAPT P10636 1/20 0.42
MAPK1 P28482 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5191096 0.77 ALDH1A1 (0.46) ALDH1A1PKML3MBTL1MAPK1
SCHEMBL10681973 0.75 SIGMAR1 (0.55) SIGMAR1ALDH1A1MEN1KMT2APOLB
SCHEMBL5214033 0.73 SIGMAR1 (0.49) SIGMAR1POLBL3MBTL1GAA
SCHEMBL5193050 0.72 KMT2A (0.41) ALDH1A1HTTPKMMEN1KMT2A
SCHEMBL22790774 0.71 ALDH1A1 (0.68) SIGMAR1ALDH1A1MEN1KMT2APOLB
SCHEMBL5195061 0.70 SIGMAR1 (0.49) SIGMAR1ALDH1A1PKMMEN1KMT2A
SCHEMBL26024178 0.70 RORC (0.51) SIGMAR1ALDH1A1HTTPKMMEN1
SCHEMBL5199484 0.69 MAPT (0.51) PKMMEN1KMT2APOLBMAPT
SCHEMBL5191582 0.69 TP53 (0.56) PKMMEN1KMT2APOLBMAPT
SCHEMBL26024193 0.69 SIGMAR1 (0.54) SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0968206-B8 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX INC (US) 2007-01-24 EP disclosed
EP-0968206-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 2000-01-05 EP disclosed
WO-1998037079-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 1998-08-27 WO disclosed