SCHEMBL5195397

SCHEMBL5195397

CN1CCN(Cc2ccc3c(c2)CCC3)C(CC(N)=O)C1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.41
FAAH O00519 1/20 0.39
DOCK5 Q9H7D0 1/20 0.38
MAPK8 P45983 2/20 0.37
KDM2B Q8NHM5 1/20 0.36
OPRD1 P41143 3/20 0.36
SMN1; SMN2 Q16637 2/20 0.35
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
HPGD P15428 1/20 0.34
CYP2C19 P33261 1/20 0.34
HRH3 Q9Y5N1 1/20 0.34
RXRB P28702 1/20 0.34
TP53 P04637 1/20 0.34
ALOX15 P16050 1/20 0.34
NTRK1 P04629 1/20 0.34
CSF1R P07333 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5214033 0.81 SIGMAR1 (0.49) SIGMAR1
SCHEMBL5208447 0.79 FAAH (0.64) FAAHSMN1; SMN2NPC1RAB9ATP53
SCHEMBL26639370 0.70 SMN1; SMN2 (0.33) SIGMAR1SMN1; SMN2
SCHEMBL25154270 0.69 SIGMAR1 (0.59) SIGMAR1
SCHEMBL25154734 0.69 SIGMAR1 (0.59) SIGMAR1
SCHEMBL14615038 0.68 CHKA (0.57) FAAH
SCHEMBL5191096 0.67 ALDH1A1 (0.46) OPRD1SMN1; SMN2
SCHEMBL658778 0.67 MAPK8 (0.55) MAPK8SMN1; SMN2CYP1A2CYP2D6HPGD
SCHEMBL31339549 0.67 MAPK8 (0.55) MAPK8SMN1; SMN2CYP1A2CYP2D6HPGD
SCHEMBL5192001 0.66 SIGMAR1 (0.56) SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0968206-B8 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX INC (US) 2007-01-24 EP disclosed
EP-0968206-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 2000-01-05 EP disclosed
WO-1998037079-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 1998-08-27 WO disclosed