SCHEMBL5196351

SCHEMBL5196351

O=C(O)C1CC(c2cnccn2)C(c2cncs2)N1

nearest known ligand 0.33

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.33
KDM4E B2RXH2 1/20 0.33
KDM1A O60341 1/20 0.31
MAPT P10636 1/20 0.31
HSD17B10 Q99714 1/20 0.31
CYP2D6 P10635 2/20 0.30
LMNA P02545 2/20 0.30
BLM P54132 2/20 0.30
ALOX15 P16050 1/20 0.30
TSHR P16473 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP2C19 P33261 1/20 0.30
RAB9A P51151 1/20 0.30
MEN1 O00255 1/20 0.30
THRB P10828 1/20 0.30
PMP22 Q01453 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6633848 0.84 KDM4E (0.32) ALDH1A1KDM4E
SCHEMBL6634950 0.82 KDM4E (0.34) ALDH1A1KDM4EMAPTHSD17B10CYP2D6
SCHEMBL6633356 0.78 KDM4E (0.37) ALDH1A1KDM4EMAPTHSD17B10CYP2D6
SCHEMBL6636875 0.75 CYP19A1 (0.42) ALDH1A1KDM4EMAPTLMNARAB9A
SCHEMBL5217655 0.74 TBXAS1 (0.31)
SCHEMBL6632885 0.73 HTT (0.41) ALDH1A1KDM4EHSD17B10LMNATSHR
SCHEMBL1667203 0.67 KDM4E (0.41) KDM4ETSHR
SCHEMBL31076264 0.67 KDM4E (0.41) KDM4ETSHR
SCHEMBL1667202 0.67 KDM4E (0.41) KDM4ETSHR
Hydrochloric Acid SCHEMBL2521887 0.66 KDM4E (0.40) KDM4ETSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1812431-A1 4-(PYRAZINE-2-YL)-PYRROLIDINE-2-CARBOXYLIC ACID COMPOUNDS AND DERIVATIVES THEREOF AS HEPATITIS C VIRUS INHIBITORS GLAXO GROUP LIMITED (GB) 2007-08-01 EP disclosed
WO-2007039145-A1 C (2) -HETEROARYLMETHYL-C (4) -PYRAZINYL-2-YL ACYL PYRROLIDINE COMPOUNDS AND THEIR USE FOR TREATING VIRAL INFECTIONS, ESPECIALLY HEPATITIS C VIRUS GLAXO GROUP LIMITED (GB) 2007-04-12 WO disclosed
WO-2007039143-A1 C (2) -HETEROARYLMETHYL-C (4) -PYRAZIN-2-YL ACYL PYRROLIDINE COMPOUNDS AND THEIR USER FOR TREATING VIRAL INFECTIONS, ESPECIALLY HEPATITICS C (HCV) GLAXO GROUP LIMITED (GB) 2007-04-12 WO disclosed
WO-2006045615-A1 4- (PYRAZINE-2-YL) -PYRROLIDINE-2-CARBOXYLIC ACID COMPOUNDS AND DERIVATIVES THEREOF AS HEPATITIS C VIRUS INHIBITORS GLAXO GROUP LIMITED (GB) 2006-05-04 WO disclosed