SCHEMBL6632885

SCHEMBL6632885

O=C(O)C1CC(c2cnccn2)C(c2nc3ccccc3s2)N1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.41
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
PKM P14618 1/20 0.41
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
ALDH1A1 P00352 3/20 0.36
UBE2M P61081 6/20 0.36
DCUN1D1 Q96GG9 6/20 0.36
LMNA P02545 3/20 0.36
TP53 P04637 2/20 0.36
POLB P06746 1/20 0.36
MAPK1 P28482 1/20 0.36
ROCK2 O75116 1/20 0.36
TSHR P16473 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
HSD17B10 Q99714 1/20 0.36
SCD O00767 1/20 0.35
KDM4E B2RXH2 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6633356 0.80 KDM4E (0.37) RAB9ASMN1; SMN2MEN1KMT2AALDH1A1
SCHEMBL6636875 0.76 CYP19A1 (0.42) NPC1RAB9ASMN1; SMN2KMT2AALDH1A1
SCHEMBL6633848 0.74 KDM4E (0.32) ALDH1A1KDM4E
SCHEMBL5196351 0.73 ALDH1A1 (0.33) RAB9AMEN1KMT2AALDH1A1LMNA
SCHEMBL5214156 0.73 MAPT (0.36) HTTNPC1RAB9ASMN1; SMN2PKM
SCHEMBL3902204 0.68 ALDH1A1 (0.47) HTTNPC1RAB9ASMN1; SMN2PKM
SCHEMBL907510 0.63 KMT2A (0.51) HTTSMN1; SMN2MEN1KMT2AALDH1A1
SCHEMBL1667203 0.63 KDM4E (0.41) TSHRKDM4E
SCHEMBL31076264 0.63 KDM4E (0.41) TSHRKDM4E
SCHEMBL1667202 0.63 KDM4E (0.41) TSHRKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1440069-A1 4-(6-MEMBERED)-HETEROARYL ACYL PYRROLIDINE DERIVATIVES AS HCV INHIBITORS GLAXO GROUP LIMITED (GB) 2004-07-28 EP disclosed
WO-2003037895-A1 4-(6-MEMBERED)-HETEROARYL ACYL PYRROLIDINE DERIVATIVES AS HCV INHIBITORS GLAXO GROUP LIMITED (GB) 2003-05-08 WO disclosed