SCHEMBL6633356

SCHEMBL6633356

O=C(O)C1CC(c2cnccn2)C(c2ccccn2)N1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.37
ALDH1A1 P00352 3/20 0.37
CYP2A6 P11509 1/20 0.34
ESR1 P03372 1/20 0.34
PABPC1 P11940 1/20 0.34
PLK1 P53350 1/20 0.34
METAP2 P50579 1/20 0.33
HSD17B10 Q99714 3/20 0.33
MAPT P10636 2/20 0.33
MEN1 O00255 2/20 0.33
THRB P10828 2/20 0.33
ALOX15 P16050 2/20 0.33
KMT2A Q03164 2/20 0.33
POLB P06746 1/20 0.33
HPGD P15428 1/20 0.33
MAPK1 P28482 1/20 0.33
CASP1 P29466 1/20 0.33
BRCA1 P38398 1/20 0.33
CASP7 P55210 1/20 0.33
TDP1 Q9NUW8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6636875 0.81 CYP19A1 (0.42) KDM4EALDH1A1MAPTKMT2ASMN1; SMN2
SCHEMBL6632885 0.80 HTT (0.41) KDM4EALDH1A1HSD17B10MEN1KMT2A
SCHEMBL5196351 0.78 ALDH1A1 (0.33) KDM4EALDH1A1HSD17B10MAPTMEN1
SCHEMBL6633848 0.76 KDM4E (0.32) KDM4EALDH1A1
SCHEMBL8871412 0.72 P4HTM (0.35) KDM4EALDH1A1ESR1PABPC1PLK1
SCHEMBL1667202 0.69 KDM4E (0.41) KDM4EPABPC1TSHR
SCHEMBL31076264 0.69 KDM4E (0.41) KDM4EPABPC1TSHR
SCHEMBL1667203 0.69 KDM4E (0.41) KDM4EPABPC1TSHR
SCHEMBL3831051 0.68 ALDH1A1 (0.60) KDM4EALDH1A1HSD17B10MAPTMEN1
SCHEMBL3831047 0.68 ALDH1A1 (0.60) KDM4EALDH1A1HSD17B10MAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1440069-A1 4-(6-MEMBERED)-HETEROARYL ACYL PYRROLIDINE DERIVATIVES AS HCV INHIBITORS GLAXO GROUP LIMITED (GB) 2004-07-28 EP disclosed
WO-2003037895-A1 4-(6-MEMBERED)-HETEROARYL ACYL PYRROLIDINE DERIVATIVES AS HCV INHIBITORS GLAXO GROUP LIMITED (GB) 2003-05-08 WO disclosed