SCHEMBL5198822

SCHEMBL5198822

CCC(C)OP(=O)(O)COc1ccc(C(=O)Cl)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 3/20 0.39
HPGD P15428 1/20 0.39
PLK1 P53350 2/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
ADRB2 P07550 1/20 0.36
ADRB3 P13945 1/20 0.36
PARP10 Q53GL7 1/20 0.36
MAPK1 P28482 1/20 0.35
TAS1R3 Q7RTX0 1/20 0.35
TAS1R1 Q7RTX1 1/20 0.35
TSHR P16473 2/20 0.35
NPC1 O15118 2/20 0.35
RAB9A P51151 1/20 0.35
ALDH1A1 P00352 1/20 0.35
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
BLM P54132 1/20 0.34
LMNA P02545 1/20 0.34
POLB P06746 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4169306 0.88 MAPT (0.48) NPSR1HPGDRAB9AALDH1A1LMNA
SCHEMBL4172471 0.82 KDM4E (0.43) MEN1KMT2AADRB2ADRB3MAPK1
SCHEMBL9055592 0.81 CYP2C9 (0.54) CYP2C9CYP2C19LMNAMAPT
SCHEMBL3187016 0.80 ALDH1A1 (0.43) HPGDMEN1KMT2AADRB2ADRB3
SCHEMBL8727337 0.77 TAAR1 (0.41) ADRB2ADRB3
SCHEMBL8681272 0.75 KMT2A (0.46) KMT2APARP10ALDH1A1POLBMAPT
SCHEMBL4167588 0.73 FDPS (0.44) MEN1KMT2AADRB2LMNAPOLB
SCHEMBL4156218 0.73 CHRNB2 (0.41) ADRB2ADRB3MAPK1CYP2C9CYP2C19
SCHEMBL5198811 0.73 PLK1 (0.45) NPSR1HPGDPLK1KMT2APARP10
SCHEMBL1251493 0.71 ADRB2 (0.33) ADRB2ADRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1809299-A2 PHOSPHONATE SUBSTITUTED KINASE INHIBITORS GILEAD SCIENCES, INC. (US) 2007-07-25 EP disclosed
WO-2006047507-A2 PHOSPHONATE SUBSTITUTED KINASE INHIBITORS GILEAD SCIENCES, INC. (US) 2006-05-04 WO disclosed