SCHEMBL5201

SCHEMBL5201

Fc1ccc(C[Zn]Br)cc1

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 5/20 0.48
LOXL2 Q9Y4K0 1/20 0.48
TAAR1 Q96RJ0 3/20 0.44
AGXT P21549 2/20 0.42
PLA2G1B P04054 1/20 0.38
ATG4B Q9Y4P1 1/20 0.38
MAOB P27338 1/20 0.38
MIF P14174 1/20 0.38
LMNA P02545 1/20 0.38
AOC3 Q16853 1/20 0.37
CHRM2 P08172 1/20 0.37
TRPA1 O75762 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3297380 0.77 TAAR1 (0.50) IDO1LOXL2TAAR1AGXTMAOB
SCHEMBL20745628 0.77 IDO1 (0.52) IDO1LOXL2TAAR1AGXTPLA2G1B
SCHEMBL3304004 0.76 IDO1 (0.41) IDO1TAAR1AGXT
SCHEMBL1980351 0.74 CYP2A6 (0.47) IDO1TAAR1
SCHEMBL2217320 0.72 IDO1 (0.48) IDO1LOXL2TAAR1AGXTPLA2G1B
SCHEMBL852178 0.72 IDO1 (0.48) IDO1LOXL2TAAR1AGXTPLA2G1B
SCHEMBL4176273 0.72 CYP3A4 (0.42) IDO1
SCHEMBL1444597 0.72 IDO1 (0.48) IDO1TAAR1AGXTMAOBLMNA
SCHEMBL4924208 0.72 IDO1 (0.48) IDO1TAAR1AGXTLMNACHRM2
SCHEMBL158407 0.72 TP53 (0.46) IDO1TAAR1LMNATRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 54 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250353856-A1 COMPOUND ACTIVE AS INHIBITOR OF COLONY STIMULATION FACTOR-1 RECEPTOR (CSF-1R) NORWEGIAN UNIV SCI & TECH NTNU (NO) 2025-11-20 US disclosed
EP-4578856-A1 HETEROCYCLIC COMPOUND Ubience Inc. (JP) 2025-07-02 EP disclosed
WO-2024079342-A1 COMPOUND ACTIVE AS INHIBITOR OF COLONY STIMULATION FACTOR-1 RECEPTOR (CSF-1R) NORWEGIAN UNIVERSITY OF SCIENCE AND TECHNOLOGY (NTNU) (NO) 2024-04-18 WO disclosed
WO-2024071371-A1 HETEROCYCLIC COMPOUND ユビエンス株式会社 2024-04-04 WO disclosed
US-11608339-B2 5-HT2C receptor agonists and compositions and methods of use ARENA PHARMACEUTICALS, INC. (US) 2023-03-21 US disclosed
EP-3500570-B1 5-HT2C RECEPTOR AGONISTS AND COMPOSITIONS AND METHODS OF USE ARENA PHARM INC (US) 2022-10-05 EP disclosed
US-20210214355-A1 5-HT2C RECEPTOR AGONISTS AND COMPOSITIONS AND METHODS OF USE ARENA PHARMACEUTICALS, INC. 2021-07-15 US disclosed
US-10836764-B2 5-HT2C receptor agonists and compositions and methods of use ARENA PHARMACEUTICALS, INC. (US) 2020-11-17 US disclosed
US-20190225612-A1 5-HT2C RECEPTOR AGONISTS AND COMPOSITIONS AND METHODS OF USE ARENA PHARMACEUTICALS, INC. 2019-07-25 US disclosed
US-10000456-B2 Polycyclic compounds as lysophosphatidic acid receptor antagonists AMIRA PHARMACEUTICALS, INC. (US) 2018-06-19 US disclosed
WO-2005042491-A1 BENZAZEPINE DERIVATIVES AND METHODS OF PROPHYLAXIS OR TREATMENT OF 5HT2C RECEPTOR ASSOCIATED DISEASES ARENA PHARMACEUTICALS, INC. (US) 2005-05-12 WO disclosed
US-20040229909-A1 Antiviral agent SHIONOGI & CO., LTD. (JP) 2004-11-18 US disclosed
US-20040116479-A1 Method of inhibiting angiogenesis ABBOTT LABORATORIES 2004-06-17 US disclosed
WO-2004032908-A9 METHOD OF INHIBITING ANGIOGENESIS ABBOTT LAB (US) 2004-05-27 WO disclosed
EP-1422218-A1 ANTIVIRAL AGENT SHIONOGI & CO., LTD. (JP) 2004-05-26 EP disclosed
WO-2004032908-A2 METHOD OF INHIBITING ANGIOGENESIS ABBOTT LABORATORIES (US) 2004-04-22 WO disclosed
US-20040067985-A1 Method of inhibiting angiogenesis ABBOT LABORATORIES 2004-04-08 US disclosed
US-5580989-A Process for the preparation of N-4-[(substituted phenyl)alkylheterocyclic]-N ABBOTT LABORATORIES (US) 1996-12-03 US disclosed
EP-0726897-A1 PROCESS FOR THE PREPARATION OF N-4- (SUBSTITUTED PHENYL)ALKYLTHIENYL]-, AND N-4- (SUBSTITUTED PHENYL)ALKYLFURYL]BUT-3-YN-2-YL]-N-HYDROXYUREA COMPOUNDS Abbott Laboratories (US) 1996-08-21 EP disclosed
WO-1995012589-A1 PROCESS FOR THE PREPARATION OF N-4-[(SUBSTITUTED PHENYL)ALKYLTHIENYL]-, AND N-4-[(SUBSTITUTED PHENYL)ALKYLFURYL]BUT-3-YN-2-YL]-N-HYDROXYUREA COMPOUNDS ABBOTT LABORATORIES (US) 1995-05-11 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190225612-A1 5-HT2C RECEPTOR AGONISTS AND COMPOSITIONS AND METHODS OF USE HTR2C, HTR2A, TPH2 IDO1 157/4885LOXL2 678/4885TAAR1 55/4885
US-11608339-B2 5-HT2C receptor agonists and compositions and methods of use HTR2C, HTR2A, TPH2 IDO1 275/4885LOXL2 477/4885TAAR1 76/4885
US-20040229909-A1 Antiviral agent ZC3HAV1, ZC3HAV1L, DUT IDO1 78/4885LOXL2 2766/4885TAAR1 4395/4885
US-20040067985-A1 Method of inhibiting angiogenesis VEGFA, PGF, FLT4 IDO1 2042/4885LOXL2 660/4885TAAR1 4748/4885
US-20210214355-A1 5-HT2C RECEPTOR AGONISTS AND COMPOSITIONS AND METHODS OF USE HTR2C, HTR2A, TPH2 IDO1 219/4885LOXL2 871/4885TAAR1 54/4885
US-10000456-B2 Polycyclic compounds as lysophosphatidic acid receptor antagonists LPAR1, LPAR2, LPAR4 IDO1 3172/4885LOXL2 96/4885TAAR1 397/4885
US-20250353856-A1 COMPOUND ACTIVE AS INHIBITOR OF COLONY STIMULATION FACTOR-1 RECEPTOR (CSF-1R) CSF1R, CSF3R, IL1RN IDO1 1572/4885LOXL2 3647/4885TAAR1 437/4885
US-10836764-B2 5-HT2C receptor agonists and compositions and methods of use HTR2C, HTR2A, TPH2 IDO1 275/4885LOXL2 477/4885TAAR1 76/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.