SCHEMBL5201261

SCHEMBL5201261

Cc1ccc(CC2=NCCN2)c(C)c1NS(C)(=O)=O

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 8/20 0.59
HTR1B P28222 7/20 0.59
ADRA1A P35348 8/20 0.52
ADRA2A P08913 6/20 0.48
ADRA2C P18825 6/20 0.48
ADRA1D P25100 5/20 0.48
ADRA1B P35368 5/20 0.48
ADRA2B P18089 3/20 0.48
TAAR1 Q96RJ0 3/20 0.45
NR3C1 P04150 1/20 0.41
RAD52 P43351 1/20 0.40
LMNA P02545 2/20 0.39
HTR1A P08908 2/20 0.39
CYP2D6 P10635 2/20 0.39
MAPK1 P28482 2/20 0.39
MAPT P10636 1/20 0.39
OPRM1 P35372 1/20 0.39
NISCH Q9Y2I1 1/20 0.39
TP53 P04637 1/20 0.39
CHRM2 P08172 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5203869 0.99 HTR1D (0.57) HTR1DHTR1BADRA1AADRA2AADRA2C
SCHEMBL4986530 0.81 ADRA1A (0.50) HTR1DHTR1BADRA1AADRA2AADRA2C
SCHEMBL2561416 0.81 HTR1D (0.50) HTR1DHTR1BADRA1AADRA2AADRA2C
SCHEMBL4992395 0.81 HTR1D (0.50) HTR1DHTR1BADRA1AADRA2AADRA2C
SCHEMBL13752307 0.81 HTR1D (0.50) HTR1DHTR1BADRA1AADRA2AADRA2C
SCHEMBL5200657 0.80 TAAR1 (0.52) HTR1DHTR1BADRA1AADRA2AADRA2C
Hydrochloric Acid SCHEMBL3726850 0.80 HTR1D (0.49) HTR1DHTR1BADRA1AADRA2AADRA2C
SCHEMBL5201030 0.80 ADRA1A (0.80) ADRA1AADRA2AADRA2CADRA1DADRA1B
Hydrochloric Acid SCHEMBL5203075 0.79 TAAR1 (0.51) HTR1DHTR1BADRA1AADRA2AADRA2C
SCHEMBL4993251 0.79 HTR1B (0.48) HTR1DHTR1BADRA1AADRA2AADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0887346-B1 N-Phenyl-alkylsulfonamide derivatives, their preparation and their use as alpha1A/1L adrenoceptor agonists HOFFMANN LA ROCHE (CH) 2007-12-12 EP disclosed