SCHEMBL5201332

SCHEMBL5201332

CCOC(=O)Cc1ccc(CC(=O)OCC)c(N)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.50
GAA P10253 1/20 0.50
GFER P55789 1/20 0.50
CYP4Z1 Q86W10 1/20 0.44
SMN1; SMN2 Q16637 3/20 0.44
PKM P14618 2/20 0.44
NPC1 O15118 1/20 0.44
NFKB1 P19838 1/20 0.44
RAB9A P51151 1/20 0.44
NFKB2 Q00653 1/20 0.44
RELA Q04206 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
MAPT P10636 2/20 0.43
CYP4F2 P78329 1/20 0.41
CYP4A11 Q02928 1/20 0.41
PPIB P23284 1/20 0.41
PPIA P62937 1/20 0.41
PPID Q08752 1/20 0.41
PPIG Q13427 1/20 0.41
CHEK1 O14757 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5100488 0.95 ALDH1A1 (0.51) ALDH1A1GAAGFERCYP4Z1SMN1; SMN2
SCHEMBL5201334 0.92 GAA (0.43) ALDH1A1GAAGFERCYP4Z1SMN1; SMN2
SCHEMBL25879759 0.91 CYP4F2 (0.43) ALDH1A1GAAGFERCYP4Z1SMN1; SMN2
SCHEMBL31287243 0.87 ALDH1A1 (0.53) ALDH1A1GAAGFERCYP4Z1SMN1; SMN2
SCHEMBL118588 0.87 ALDH1A1 (0.53) ALDH1A1GAAGFERCYP4Z1SMN1; SMN2
SCHEMBL2131319 0.85 LMNA (0.46) ALDH1A1SMN1; SMN2PKMMAPTPPIB
SCHEMBL21437852 0.85 NLRP3 (0.43) ALDH1A1GAASMN1; SMN2PKMNPC1
SCHEMBL4278414 0.84 ALDH1A1 (0.50) ALDH1A1GAAGFERCYP4Z1SMN1; SMN2
SCHEMBL5656071 0.84 ALDH1A1 (0.71) ALDH1A1GAAGFERCYP4Z1SMN1; SMN2
SCHEMBL20383846 0.84 PKM (0.42) ALDH1A1SMN1; SMN2PKMCHEK1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1179532-B1 PROCESS FOR THE PRODUCTION OF INDOLE DERIVATIVES AND INTERMEDIATES THEREFOR EISAI R&D MAN CO LTD (JP) 2007-06-13 EP disclosed
US-6573384-B1 1,4-substituted cyclic amine compound which is useful as a pharmaceutical, and an intermediate for the process EISAI CO., LTD. (JP) 2003-06-03 US disclosed
EP-1179532-A1 PROCESS FOR THE PRODUCTION OF INDOLE DERIVATIVES AND INTERMEDIATES THEREFOR Eisai Co., Ltd. (JP) 2002-02-13 EP disclosed