SCHEMBL5201374

SCHEMBL5201374

CCCCOC(=O)NC(Cc1nccs1)C(=O)OC

nearest known ligand 0.55

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.55
CTSK P43235 4/20 0.46
PKM P14618 2/20 0.43
MAPK1 P28482 2/20 0.41
TSHR P16473 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
CYP3A4 P08684 3/20 0.40
RAB9A P51151 1/20 0.39
HRH2 P25021 1/20 0.39
HRH1 P35367 1/20 0.39
ALDH1A1 P00352 2/20 0.39
FDPS P14324 1/20 0.38
ITGB3 P05106 1/20 0.38
ITGA2B P08514 1/20 0.38
HSPA5 P11021 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6207414 0.91 L3MBTL1 (0.55) L3MBTL1CTSKPKMMAPK1TSHR
SCHEMBL5924778 0.81 CTSK (0.44) CTSKCYP3A4FDPSITGB3ITGA2B
SCHEMBL2398131 0.81 CTSK (0.44) CTSKCYP3A4FDPSITGB3ITGA2B
SCHEMBL4385669 0.74 POLB (0.62) L3MBTL1CTSKTSHRRAB9AALDH1A1
SCHEMBL3652453 0.74 POLB (0.62) L3MBTL1CTSKTSHRRAB9AALDH1A1
SCHEMBL5201378 0.73 L3MBTL1 (0.54) L3MBTL1CTSKPKMMAPK1TSHR
SCHEMBL1696818 0.73 CA1 (0.46) L3MBTL1MAPK1SMN1; SMN2RAB9AALDH1A1
SCHEMBL20683487 0.73 CA1 (0.46) L3MBTL1MAPK1SMN1; SMN2RAB9AALDH1A1
SCHEMBL8008631 0.73 NPSR1 (0.53) MAPK1TSHRSMN1; SMN2ALDH1A1
SCHEMBL6826832 0.73 NPSR1 (0.53) MAPK1TSHRSMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1817275-A1 HALOALKYL CONTAINING COMPOUNDS AS CYSTEINE PROTEASE INHIBITORS Schering Aktiengesellschaft (DE) 2007-08-15 EP disclosed
WO-2006060494-A1 HALOALKYL CONTAINING COMPOUNDS AS CYSTEINE PROTEASE INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 2006-06-08 WO disclosed