SCHEMBL8985906

SCHEMBL8985906

O=C(Nc1ccc2[nH]c(C(=O)O)cc2c1)OCc1ccccc1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRD5A2 P31213 3/20 0.60
ALDH1A1 P00352 2/20 0.60
KDM4E B2RXH2 2/20 0.60
HPGD P15428 2/20 0.60
HSD17B10 Q99714 2/20 0.60
CYP1A2 P05177 1/20 0.60
CYP2C9 P11712 1/20 0.60
ROCK2 O75116 2/20 0.57
MGLL Q99685 2/20 0.54
MAPT P10636 3/20 0.52
TP53 P04637 2/20 0.52
NPC1 O15118 1/20 0.52
TSHR P16473 1/20 0.52
RAB9A P51151 1/20 0.52
ATM Q13315 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
POLB P06746 1/20 0.50
SRD5A1 P18405 1/20 0.50
ENPP2 Q13822 2/20 0.49
MMP13 P45452 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8985820 0.88 MMP13 (0.68) ALDH1A1KDM4EHPGDHSD17B10ROCK2
SCHEMBL9687922 0.86 SRD5A2 (0.46) SRD5A2ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL5200855 0.84 MGLL (0.60) ALDH1A1ROCK2MGLLMAPTTP53
SCHEMBL9688119 0.82 MMP13 (0.61) ALDH1A1KDM4EHPGDHSD17B10ROCK2
SCHEMBL9127299 0.82 NPC1 (0.67) ALDH1A1KDM4ENPC1RAB9ASMN1; SMN2
SCHEMBL7833243 0.81 LEF1 (0.55) SRD5A2ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL7908588 0.80 KCNQ2 (0.57) ALDH1A1ROCK2MGLLMAPTTP53
SCHEMBL28365377 0.80 EPHX2 (0.57) SRD5A2ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL4432278 0.79 MGLL (0.65) ALDH1A1KDM4ECYP1A2ROCK2MGLL
SCHEMBL30207797 0.79 MGLL (0.65) ALDH1A1KDM4ECYP1A2ROCK2MGLL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5563142-A INHIBITORS OF VIRAL REVERSE TRANSCRIPTASE THE UPJOHN COMPANY (US) 1996-10-08 US disclosed
EP-0507861-B1 DIAROMATIC SUBSTITUTED ANTI-AIDS COMPOUNDS UPJOHN CO (US) 1996-09-11 EP disclosed
US-5489593-A Anti-aids piperazines THE UPJOHN COMPANY (US) 1996-02-06 US disclosed
EP-0507861-A1 DIAROMATIC SUBSTITUTED ANTI-AIDS COMPOUNDS. UPJOHN CO (US) 1992-10-14 EP disclosed
WO-1991009849-A1 DIAROMATIC SUBSTITUTED ANTI-AIDS COMPOUNDS THE UPJOHN COMPANY (US) 1991-07-11 WO disclosed