SCHEMBL5202866

SCHEMBL5202866

CCOc1ccc(N2CCC(n3c(Cl)cc4ccc(CC(=O)O)cc43)CC2)c(F)c1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ACACB O00763 5/20 0.41
PTGER4 P35408 2/20 0.38
FFAR1 O14842 5/20 0.37
NPY2R P49146 1/20 0.36
GAA P10253 2/20 0.36
PTGDR2 Q9Y5Y4 1/20 0.35
HPGD P15428 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
CHRM4 P08173 1/20 0.34
PTGS1 P23219 1/20 0.34
AKR1C3 P42330 1/20 0.34
AKR1C2 P52895 1/20 0.34
HTR2A P28223 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5205007 0.77 ACACB (0.42) ACACBPTGER4FFAR1NPY2RGAA
SCHEMBL5204378 0.75 ACACB (0.42) ACACBNPY2RGAAHPGDSMN1; SMN2
SCHEMBL5206812 0.73 SIGMAR1 (0.40) PTGDR2HTR2A
SCHEMBL5205196 0.72 HTR2A (0.47) HTR2A
SCHEMBL5201290 0.71 ACACB (0.44) ACACBPTGER4FFAR1NPY2RPTGDR2
SCHEMBL5201956 0.70 KCNH2 (0.43) HTR2A
SCHEMBL5206818 0.70 KDM4E (0.36) PTGDR2HPGD
SCHEMBL5206821 0.69 KDM4E (0.37) HPGD
SCHEMBL4137101 0.68 L3MBTL1 (0.54) ACACBNPY2RHPGDSMN1; SMN2
SCHEMBL5206815 0.67 SLC22A12 (0.44) SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1179532-B1 PROCESS FOR THE PRODUCTION OF INDOLE DERIVATIVES AND INTERMEDIATES THEREFOR EISAI R&D MAN CO LTD (JP) 2007-06-13 EP disclosed
US-6573384-B1 1,4-substituted cyclic amine compound which is useful as a pharmaceutical, and an intermediate for the process EISAI CO., LTD. (JP) 2003-06-03 US disclosed
EP-1179532-A1 PROCESS FOR THE PRODUCTION OF INDOLE DERIVATIVES AND INTERMEDIATES THEREFOR Eisai Co., Ltd. (JP) 2002-02-13 EP disclosed