SCHEMBL5201290

SCHEMBL5201290

CCOC(=O)Cc1ccc(CC(=O)O)cc1NC1CCN(c2ccc(OCC)cc2F)CC1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACACB O00763 4/20 0.44
NOS1 P29475 1/20 0.41
NOS2 P35228 1/20 0.41
L3MBTL1 Q9Y468 2/20 0.39
MAPT P10636 4/20 0.39
NPC1 O15118 1/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
HPGD P15428 1/20 0.39
ALOX15 P16050 1/20 0.39
TSHR P16473 1/20 0.39
MAPK1 P28482 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
HSD17B10 Q99714 1/20 0.39
NPY2R P49146 1/20 0.38
PTGER4 P35408 1/20 0.38
FFAR1 O14842 1/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
PTGDR2 Q9Y5Y4 3/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5201976 0.79 OPRM1 (0.43) ALDH1A1HSD17B10PTGDR2POLBKDM1A
SCHEMBL5201971 0.74 CACNA1G (0.44) L3MBTL1ALDH1A1MAPK1NPSR1HSD17B10
SCHEMBL5205007 0.72 ACACB (0.42) ACACBHPGDNPY2RPTGER4FFAR1
SCHEMBL5202266 0.71 CACNA1G (0.42) ALDH1A1HSD17B10KDM1AHTR2A
SCHEMBL5202866 0.71 ACACB (0.41) ACACBHPGDNPY2RPTGER4FFAR1
SCHEMBL4137101 0.69 L3MBTL1 (0.54) ACACBL3MBTL1MAPTNPC1ALDH1A1
SCHEMBL20521460 0.68 TSHR (0.55) L3MBTL1MAPTNPC1ALDH1A1LMNA
SCHEMBL5203925 0.68 CNR1 (0.43) L3MBTL1ALDH1A1TSHRMAPK1HSD17B10
SCHEMBL5201178 0.67 ALDH1A1 (0.44) MAPTALDH1A1TSHRHSD17B10
SCHEMBL31341914 0.67 PANK3 (0.43) ACACBL3MBTL1MAPTALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1179532-B1 PROCESS FOR THE PRODUCTION OF INDOLE DERIVATIVES AND INTERMEDIATES THEREFOR EISAI R&D MAN CO LTD (JP) 2007-06-13 EP disclosed
US-6573384-B1 1,4-substituted cyclic amine compound which is useful as a pharmaceutical, and an intermediate for the process EISAI CO., LTD. (JP) 2003-06-03 US disclosed
EP-1179532-A1 PROCESS FOR THE PRODUCTION OF INDOLE DERIVATIVES AND INTERMEDIATES THEREFOR Eisai Co., Ltd. (JP) 2002-02-13 EP disclosed