SCHEMBL5202929

SCHEMBL5202929

COc1cccc(Cn2cc(C3CCN(C(=O)c4c(-c5ccccc5Cl)noc4C)C3)c3ccccc32)c1

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.51
MEN1 O00255 2/20 0.51
LMNA P02545 6/20 0.46
ALDH1A1 P00352 4/20 0.46
HTT P42858 2/20 0.46
NPC1 O15118 1/20 0.46
GAA P10253 2/20 0.46
TSHR P16473 4/20 0.46
MAPK1 P28482 1/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
EPAS1 Q99814 1/20 0.46
GPBAR1 Q8TDU6 1/20 0.45
USP2 O75604 1/20 0.44
PKM P14618 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
KDM4E B2RXH2 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5203496 0.85 KMT2A (0.60) KMT2AMEN1LMNAALDH1A1HTT
SCHEMBL5202293 0.79 THRB (0.49) KMT2AMEN1LMNAALDH1A1KDM4E
SCHEMBL5282265 0.79 HCRTR1 (0.39) KMT2AMEN1LMNAALDH1A1HTT
SCHEMBL5204484 0.79 SLC2A1 (0.47) LMNAALDH1A1HTTNPSR1
SCHEMBL5203382 0.78 MAPT (0.46) KMT2AMEN1LMNAALDH1A1SMN1; SMN2
SCHEMBL4852934 0.77 HRH2 (0.50) KMT2ALMNAALDH1A1HTTNPC1
SCHEMBL5204486 0.76 MAPT (0.54) KMT2AMEN1LMNAALDH1A1HTT
SCHEMBL4858756 0.76 SLC2A1 (0.49) KMT2AMEN1LMNAALDH1A1HTT
SCHEMBL5205779 0.75 HRH2 (0.49) LMNAALDH1A1HTTTSHRSMN1; SMN2
SCHEMBL5203370 0.75 HRH2 (0.47) LMNAALDH1A1HTTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1654253-B1 SUBSTITUTED 3-PYRROLIDIN-INDOLE DERIVATIVES GRUENENTHAL GMBH (DE) 2007-01-03 EP claimed