SCHEMBL5282265

SCHEMBL5282265

COc1cccc(CN2OC(C)=C(C(=O)C3C(c4cn(Cc5cccc(OC)c5)c5ccccc45)CCN3C(=O)c3c(-c4ccccc4Cl)noc3C)C2c2ccccc2Cl)c1

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 4/20 0.39
HCRTR2 O43614 3/20 0.39
TSHR P16473 4/20 0.39
GPBAR1 Q8TDU6 2/20 0.39
LMNA P02545 4/20 0.38
NPSR1 Q6W5P4 1/20 0.38
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
GAA P10253 2/20 0.37
ALDH1A1 P00352 2/20 0.37
HTT P42858 1/20 0.37
MAPK1 P28482 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.36
EPAS1 Q99814 1/20 0.36
MAPT P10636 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5202929 0.79 KMT2A (0.51) TSHRGPBAR1LMNANPSR1MEN1
SCHEMBL5231721 0.77 TSHR (0.51) HCRTR1HCRTR2TSHRLMNAMEN1
SCHEMBL5203496 0.65 KMT2A (0.60) TSHRLMNAMEN1KMT2AGAA
SCHEMBL4857642 0.64 MAPT (0.41) HCRTR1HCRTR2TSHRMEN1KMT2A
SCHEMBL13732613 0.63 ALDH1A1 (0.84) TSHRGPBAR1LMNAMEN1KMT2A
Hydrochloric Acid SCHEMBL13733351 0.63 ALDH1A1 (0.82) TSHRGPBAR1LMNAMEN1KMT2A
SCHEMBL5202293 0.60 THRB (0.49) LMNAMEN1KMT2AALDH1A1MAPT
SCHEMBL24480171 0.59 LMNA (0.53) LMNAALDH1A1SMN1; SMN2MAPT
SCHEMBL5204486 0.59 MAPT (0.54) TSHRLMNANPSR1MEN1KMT2A
SCHEMBL5432012 0.59 ALDH1A1 (0.44) LMNAMEN1KMT2AALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1654253-B1 SUBSTITUTED 3-PYRROLIDIN-INDOLE DERIVATIVES GRUENENTHAL GMBH (DE) 2007-01-03 EP disclosed