SCHEMBL5203380

SCHEMBL5203380

CC(c1ccc(Cl)cc1)C(CNC(=O)C1(c2cccc(Cl)c2)CCCCC1)c1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 4/20 0.42
HTRA1 Q92743 1/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
KCNH2 Q12809 2/20 0.41
IDO1 P14902 1/20 0.41
HTT P42858 1/20 0.41
TRPA1 O75762 4/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C8 P10632 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
ERCC1 P07992 1/20 0.41
ERCC4 Q92889 1/20 0.41
NPSR1 Q6W5P4 2/20 0.41
LMNA P02545 2/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
TP53 P04637 1/20 0.39
CNR1 P21554 2/20 0.38
CNR2 P34972 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5200569 0.88 TRPA1 (0.46) HDAC4SMN1; SMN2KCNH2HTTTRPA1
SCHEMBL5200440 0.85 ALDH1A1 (0.48) HDAC4SMN1; SMN2KCNH2IDO1HTT
SCHEMBL4829758 0.80 CNR1 (0.55) CNR1CNR2
SCHEMBL5202615 0.80 ALDH1A1 (0.43) TRPA1LMNATP53CNR1TSHR
SCHEMBL5205537 0.80 HDAC4 (0.42) HDAC4SMN1; SMN2TRPA1NPSR1LMNA
SCHEMBL5202867 0.79 CNR1 (0.45) HDAC4TRPA1CNR1CNR2
SCHEMBL5201399 0.78 TRPA1 (0.46) HDAC4TRPA1CNR1CNR2
SCHEMBL5201238 0.77 ITGB1 (0.45) SMN1; SMN2CNR1SLC6A2SLC6A4SLC6A3
SCHEMBL5203142 0.77 ALDH1A1 (0.48) HDAC4SMN1; SMN2TRPA1CNR1CNR2
SCHEMBL5202986 0.77 KMT2A (0.40) HDAC4SMN1; SMN2KCNH2LMNATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1490043-A4 SPIROCYCLIC AMIDES AS CANNABINOID RECEPTOR MODULATORS MERCK & CO INC (US) 2007-05-30 EP claimed
EP-1490043-A2 SPIROCYCLIC AMIDES AS CANNABINOID RECEPTOR MODULATORS Merck & Co., Inc. (US) 2004-12-29 EP claimed
WO-2003082190-A2 SPIROCYCLIC AMIDES AS CANNABINOID RECEPTOR MODULATORS MERCK & CO., INC. (US) 2003-10-09 WO claimed