SCHEMBL5203500

SCHEMBL5203500

COC(=O)Oc1ccc2cccc(N)c2n1

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 11/20 0.46
MTNR1B P49286 11/20 0.46
HTR3A P46098 1/20 0.39
MCHR1 Q99705 1/20 0.38
ALDH1A1 P00352 1/20 0.38
CFTR P13569 1/20 0.38
HSD17B10 Q99714 1/20 0.38
PARP1 P09874 1/20 0.36
PDE10A Q9Y233 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5202897 0.82 MTNR1A (0.42) MTNR1AMTNR1BHTR3AMCHR1HSD17B10
SCHEMBL3577364 0.80 MCHR1 (0.49) MTNR1AMTNR1BHTR3AMCHR1PDE10A
SCHEMBL5206188 0.79 HTR3A (0.40) HTR3AALDH1A1CFTRHSD17B10
Hydrochloric Acid SCHEMBL3583982 0.78 MCHR1 (0.47) MTNR1AMTNR1BHTR3AMCHR1PDE10A
SCHEMBL6225917 0.77 KDM4E (0.48) MTNR1AMTNR1BALDH1A1HSD17B10
SCHEMBL4707883 0.77 XIAP (0.45) MTNR1AMTNR1BMCHR1ALDH1A1CFTR
SCHEMBL4819927 0.76 ALDH1A1 (0.46) ALDH1A1CFTRHSD17B10
SCHEMBL6223869 0.73 KDM4E (0.44) MTNR1AMTNR1BALDH1A1HSD17B10
SCHEMBL11817511 0.71 KDM4E (0.56) MTNR1AMTNR1BALDH1A1HSD17B10
SCHEMBL4710517 0.71 HSD17B10 (0.33) MTNR1AMTNR1BHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1492771-B1 QUINOLINE AND ISOQUINOLINE DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF AND USE THEREOF AS ANTI-INFLAMMATORY AGENTS SCHERING AG (DE) 2007-02-28 EP disclosed
EP-1492771-A1 QUINOLINE AND ISOQUINOLINE DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF AND USE THEREOF AS ANTI-INFLAMMATORY AGENTS SCHERING AKTIENGESELLSCHAFT (DE) 2005-01-05 EP disclosed
WO-2003082827-A1 QUINOLINE AND ISOQUINOLINE DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF AND USE THEREOF AS ANTI-INFLAMMATORY AGENTS SCHERING AKTIENGESELLSCHAFT (DE) 2003-10-09 WO disclosed