SCHEMBL5203892

SCHEMBL5203892

CC(=O)Oc1ccc(Nc2nc(N)ncc2Oc2ccc(Cl)cc2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 12/20 0.46
KCNH2 Q12809 6/20 0.46
SCN5A Q14524 6/20 0.46
TTBK1 Q5TCY1 1/20 0.45
TTBK2 Q6IQ55 1/20 0.45
MAPK8 P45983 1/20 0.43
NR1I2 O75469 1/20 0.43
AHR P35869 1/20 0.43
ALDH1A1 P00352 1/20 0.42
HSP90AA1 P07900 1/20 0.42
GAA P10253 1/20 0.42
MAPT P10636 1/20 0.42
PDGFRB P09619 1/20 0.41
FLT1 P17948 1/20 0.41
KDR P35968 1/20 0.41
CCNT1 O60563 1/20 0.40
CCNC P24863 1/20 0.40
CDK8 P49336 1/20 0.40
CDK9 P50750 1/20 0.40
MEN1 O00255 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5204622 0.85 SCN9A (0.51) SCN9AKCNH2SCN5ATTBK1TTBK2
Hydrochloric Acid SCHEMBL5203439 0.84 SCN9A (0.50) SCN9AKCNH2SCN5ATTBK1TTBK2
SCHEMBL7514733 0.82 RXFP1 (0.52) SCN9AKCNH2SCN5ATTBK1TTBK2
SCHEMBL7519009 0.79 RXFP1 (0.49) SCN9AKCNH2SCN5ATTBK1TTBK2
SCHEMBL5204374 0.79 SCN9A (0.44) SCN9AKCNH2SCN5ATTBK1TTBK2
SCHEMBL5205246 0.77 SCN9A (0.45) SCN9AKCNH2SCN5ATTBK1TTBK2
SCHEMBL6481407 0.75 AURKA (0.47) SCN9AKCNH2SCN5ATTBK1TTBK2
SCHEMBL6480285 0.75 AURKA (0.53) TTBK1TTBK2ALDH1A1MAPTMEN1
SCHEMBL5207711 0.74 SCN9A (0.43) SCN9AKCNH2SCN5ATTBK1TTBK2
SCHEMBL5204470 0.74 MEN1 (0.42) SCN9AKCNH2SCN5ATTBK1TTBK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1165523-B1 NEUROTROPHIC SUBSTITUTED PYRIMIDINES KRENITSKY PHARMACEUTICALS INC (US) 2007-11-07 EP claimed
US-6916820-B1 Neurotrophic substituted pyrimidines KRENITSKY PHARMACEUTICALS, INC. (US) 2005-07-12 US claimed
EP-1165523-B1 NEUROTROPHIC SUBSTITUTED PYRIMIDINES KRENITSKY PHARMACEUTICALS INC (US) 2007-11-07 EP disclosed
US-6916820-B1 Neurotrophic substituted pyrimidines KRENITSKY PHARMACEUTICALS, INC. (US) 2005-07-12 US disclosed
EP-1165523-A1 NEUROTROPHIC SUBSTITUTED PYRIMIDINES Krenitsky Pharmaceuticals, Inc. (US) 2002-01-02 EP disclosed
WO-2000061562-A1 NEUROTROPHIC SUBSTITUTED PYRIMIDINES KRENITSKY PHARMACEUTICALS INC. (US) 2000-10-19 WO disclosed