SCHEMBL5204622

SCHEMBL5204622

Nc1ncc(Oc2ccc(Cl)cc2)c(Nc2ccc(O)cc2)n1

nearest known ligand 0.51

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 13/20 0.51
KCNH2 Q12809 6/20 0.51
SCN5A Q14524 5/20 0.51
TTBK1 Q5TCY1 2/20 0.49
TTBK2 Q6IQ55 2/20 0.49
BCL6 P41182 1/20 0.44
AURKA O14965 1/20 0.43
ADORA3 P0DMS8 1/20 0.42
SLC6A2 P23975 1/20 0.42
PDE4A P27815 1/20 0.42
KDR P35968 1/20 0.42
IKBKB O14920 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5203439 0.99 SCN9A (0.50) SCN9AKCNH2SCN5ATTBK1TTBK2
SCHEMBL6480285 0.88 AURKA (0.53) TTBK1TTBK2AURKA
SCHEMBL6472908 0.88 TTBK1 (0.43) SCN9AKCNH2SCN5ATTBK1TTBK2
SCHEMBL6481407 0.88 AURKA (0.47) SCN9AKCNH2SCN5ATTBK1TTBK2
SCHEMBL6474471 0.87 BCL6 (0.49) SCN9ASCN5ATTBK1TTBK2BCL6
SCHEMBL5204374 0.86 SCN9A (0.44) SCN9AKCNH2SCN5ATTBK1TTBK2
SCHEMBL5204470 0.86 MEN1 (0.42) SCN9AKCNH2SCN5ATTBK1TTBK2
SCHEMBL5203892 0.85 SCN9A (0.46) SCN9AKCNH2SCN5ATTBK1TTBK2
SCHEMBL6482628 0.84 BCL6 (0.44) SCN9AKCNH2SCN5ABCL6AURKA
SCHEMBL6480339 0.84 MAPT (0.44) AURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1165523-B1 NEUROTROPHIC SUBSTITUTED PYRIMIDINES KRENITSKY PHARMACEUTICALS INC (US) 2007-11-07 EP claimed
US-6916820-B1 Neurotrophic substituted pyrimidines KRENITSKY PHARMACEUTICALS, INC. (US) 2005-07-12 US claimed