SCHEMBL5210309

SCHEMBL5210309

CCOC(=O)[C@H](Cc1ccc2oc(CCCOCc3ccccc3)cc(=O)c2c1)NC(=O)OCC(C)(C)C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TYR P14679 3/20 0.41
ITGB3 P05106 2/20 0.38
ITGAV P06756 1/20 0.38
KDM4E B2RXH2 2/20 0.37
LMNA P02545 2/20 0.37
HPGD P15428 2/20 0.37
MEN1 O00255 1/20 0.37
ALDH1A1 P00352 1/20 0.37
HTT P42858 1/20 0.37
KMT2A Q03164 1/20 0.37
ITGA2B P08514 1/20 0.37
PPARG P37231 1/20 0.37
ALOX15 P16050 1/20 0.36
CASP1 P29466 1/20 0.36
HSD17B10 Q99714 1/20 0.35
POLB P06746 1/20 0.35
PPARA Q07869 1/20 0.35
ELANE P08246 1/20 0.35
TSHR P16473 1/20 0.35
CTSK P43235 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5205119 0.88 ITGB3 (0.38) TYRITGB3ITGAVKDM4ELMNA
SCHEMBL5206753 0.87 ALOX15 (0.39) TYRITGB3ITGAVKDM4ELMNA
SCHEMBL5208511 0.83 ITGB3 (0.37) TYRITGB3ITGAVKDM4ELMNA
SCHEMBL5207016 0.82 ITGB1 (0.42) TYRITGB3ITGAVKDM4ELMNA
SCHEMBL14431257 0.82 ITGB1 (0.42) TYRITGB3ITGAVKDM4ELMNA
SCHEMBL6495736 0.82 ITGB3 (0.44) TYRITGB3ITGAVITGA2BPPARG
SCHEMBL6498071 0.81 ITGB3 (0.44) TYRITGB3ITGAVMEN1KMT2A
SCHEMBL3052420 0.80 ITGB3 (0.44) TYRITGB3ITGAVITGA2BPPARG
SCHEMBL5204539 0.80 ITGB3 (0.41) ITGB3ITGAVKDM4EKMT2AITGA2B
SCHEMBL5203532 0.79 ITGB3 (0.34) TYRITGB3ITGAVKDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1124824-B1 CHROMENONE AND CHROMANONE DERIVATIVES AS INTEGRIN INHIBITORS MERCK PATENT GMBH (DE) 2007-08-22 EP disclosed