SCHEMBL5204561

SCHEMBL5204561

C[SiH](C)Oc1cc(C(C)(C)C)ccc1C=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA9 Q16790 1/20 0.39
ALDH1A1 P00352 7/20 0.39
MAPT P10636 2/20 0.38
NPSR1 Q6W5P4 2/20 0.38
MAPK1 P28482 1/20 0.38
L3MBTL1 Q9Y468 2/20 0.33
SMN1; SMN2 Q16637 3/20 0.33
TDP1 Q9NUW8 3/20 0.32
HPGD P15428 2/20 0.32
ALOX15 P16050 1/20 0.32
HSD17B10 Q99714 1/20 0.32
CYP2C19 P33261 1/20 0.32
NPC1 O15118 2/20 0.32
RAB9A P51151 2/20 0.32
PLA2G1B P04054 1/20 0.32
NFKB1 P19838 1/20 0.32
CASP3 P42574 1/20 0.32
NFKB2 Q00653 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL411850 0.83 CA1 (0.36) CA1CA2CA9ALDH1A1MAPT
SCHEMBL24398644 0.81 ALDH1A1 (0.59) CA1CA2CA9ALDH1A1MAPT
SCHEMBL31134158 0.81 ALDH1A1 (0.59) CA1CA2CA9ALDH1A1MAPT
SCHEMBL3714765 0.80 LMNA (0.35) CA1CA2CA9ALDH1A1MAPT
SCHEMBL7189375 0.80 CYP1A2 (0.40) CA1CA2CA9MAPT
SCHEMBL7189386 0.80 CYP1A2 (0.40) CA1CA2CA9MAPT
SCHEMBL4868031 0.79 CA1 (0.41) CA1CA2CA9ALDH1A1MAPT
SCHEMBL12098518 0.79 RXRA (0.46) ALDH1A1MAPTMAPK1SMN1; SMN2HPGD
SCHEMBL7366742 0.77 SCN10A (0.33) CA1CA2CA9ALDH1A1MAPT
SCHEMBL4261454 0.76 CA1 (0.31) CA1CA2CA9ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111822053-B Chiral polysulfonate diamine-metal catalyst and synthesis and application thereof 中山大学 2022-09-30 CN disclosed
CN-111822053-A Chiral polysulfonate diamine-metal catalyst and synthesis and application thereof 中山大学 2020-10-27 CN disclosed
US-7160887-B1 Aromatic amine derivatives, their production and use TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-01-09 US disclosed
CN-1834091-A Sustituted Gly derivative for treating diabetes and adiposis SHENG ZELIN (CN) 2006-09-20 CN disclosed
EP-1123918-B1 AROMATIC AMINE DERIVATIVES, PROCESS FOR THE PREPARATION THEREOF AND AGENTS CONTAINING THE SAME TAKEDA PHARMACEUTICAL (JP) 2005-03-09 EP disclosed
WO-2003024909-A1 METHOD OF PREPARING SYMMETRICAL POLYHYDROXYSTILBENES L'OREAL (FR) 2003-03-27 WO disclosed
CN-1083833-C Sulfur-substituted azetidinone compounds useful as hypocholesterolemic agents SCHERING CORP (US) 2002-05-01 CN disclosed
EP-0792264-B1 SULFUR-SUBSTITUTED AZETIDINONE COMPOUNDS USEFUL AS HYPOCHOLESTEROLEMIC AGENTS SCHERING CORP (US) 2002-02-27 EP disclosed
EP-0805132-B1 Method of producing styrene derivatives HONSHU CHEMICAL IND (JP) 2001-12-12 EP disclosed
EP-1123918-A1 AROMATIC AMINE DERIVATIVES, PROCESS FOR THE PREPARATION THEREOF AND AGENTS CONTAINING THE SAME Takeda Chemical Industries, Ltd. (JP) 2001-08-16 EP disclosed
EP-1020434-A1 3-AMIDINOANILINE DERIVATIVES, ACTIVATED BLOOD COAGULATION FACTOR X INHIBITORS, AND INTERMEDIATES FOR PRODUCING BOTH Kissei Pharmaceutical Co., Ltd. (JP) 2000-07-19 EP disclosed
US-5763560-A TREATING BENZALDEHYDE DERIVATIVE WITH ZINC AND ACTIVE CHLORIDE IN AN ORGANIC SOLVENT HONSHU CHEMICAL INDUSTRY CO., LTD. (JP) 1998-06-09 US disclosed
CN-1174548-A Sulfur-substituted azetidinone compounds useful as cholesterol lowering agents SCHERING CORP (US) 1998-02-25 CN disclosed
US-5686478-A Endothelin antagonists MERCK & CO. INC. (US) 1997-11-11 US disclosed
EP-0805132-A1 Method of producing styrene derivatives HONSHU CHEMICAL INDUSTRY CO. LTD. (JP) 1997-11-05 EP disclosed
US-5633246-A Sulfur-substituted azetidinone compounds useful as hypocholesterolemic agents SCHERING CORPORATION (US) 1997-05-27 US disclosed
US-5624920-A Sulfur-substituted azetidinone compounds useful as hypocholesterolemic agents SCHERING CORPORATION (US) 1997-04-29 US disclosed
WO-1995003295-A1 ENDOTHELIN ANTAGONISTS MERCK & CO., INC. (US) 1995-02-02 WO disclosed