SCHEMBL5205241

SCHEMBL5205241

CC(C)(C)OC(=O)NCCc1cccc(Oc2cc(Cl)ccc2N)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.46
CNR1 P21554 4/20 0.45
IDO1 P14902 2/20 0.43
TAAR1 Q96RJ0 1/20 0.41
NQO2 P16083 1/20 0.41
LMNA P02545 1/20 0.41
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
ALDH1A1 P00352 2/20 0.40
HPGD P15428 2/20 0.40
HTT P42858 2/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
TRPV1 Q8NER1 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
MAPK1 P28482 1/20 0.40
CYP2C19 P33261 1/20 0.40
CA2 P00918 1/20 0.40
TP53 P04637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5205639 0.84 LMNA (0.48) KDM4ECNR1IDO1LMNAMEN1
SCHEMBL25834083 0.81 KDM4E (0.63) KDM4ECNR1TAAR1NQO2LMNA
SCHEMBL6192699 0.80 KDM4E (0.47) KDM4ECNR1IDO1NQO2LMNA
SCHEMBL5354570 0.80 FDFT1 (0.57) IDO1NQO2
SCHEMBL5208318 0.80 HDAC1 (0.43) KDM4ECNR1TAAR1SMN1; SMN2
SCHEMBL21090366 0.79 FDFT1 (0.47) KDM4ECNR1IDO1NQO2CA2
SCHEMBL5202388 0.79 CNR1 (0.40) KDM4ECNR1MEN1KMT2AMAPT
SCHEMBL6185337 0.78 KDM4E (0.45) KDM4ECNR1IDO1TAAR1NQO2
SCHEMBL6204579 0.78 MTNR1A (0.58) CNR1TAAR1ALDH1A1HTTSMN1; SMN2
SCHEMBL6677541 0.77 CA2 (0.49) KDM4EIDO1NQO2LMNAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7160887-B1 Aromatic amine derivatives, their production and use TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-01-09 US disclosed
EP-1123918-B1 AROMATIC AMINE DERIVATIVES, PROCESS FOR THE PREPARATION THEREOF AND AGENTS CONTAINING THE SAME TAKEDA PHARMACEUTICAL (JP) 2005-03-09 EP disclosed
EP-1123918-A1 AROMATIC AMINE DERIVATIVES, PROCESS FOR THE PREPARATION THEREOF AND AGENTS CONTAINING THE SAME Takeda Chemical Industries, Ltd. (JP) 2001-08-16 EP disclosed