SCHEMBL5208318

SCHEMBL5208318

CC(C)(C)OC(=O)NCCc1cccc(Oc2cc(Cl)ccc2NCc2ccc(-c3ccccc3)cc2)c1

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.43
KDM4E B2RXH2 1/20 0.41
HIF1A Q16665 1/20 0.40
ADAMTS5 Q9UNA0 2/20 0.40
TAAR1 Q96RJ0 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
CNR1 P21554 2/20 0.39
SUCNR1 Q9BXA5 1/20 0.38
PTGDR2 Q9Y5Y4 2/20 0.38
ADRB1 P08588 1/20 0.38
ADRB3 P13945 1/20 0.38
FFAR1 O14842 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5206113 0.82 ADAMTS5 (0.48) ADAMTS5SMN1; SMN2PTGDR2FFAR1
SCHEMBL5205234 0.81 TSHR (0.46) SMN1; SMN2PTGDR2
SCHEMBL5205774 0.80 ADAMTS5 (0.40) ADAMTS5PTGDR2FFAR1
SCHEMBL5202388 0.80 CNR1 (0.40) HDAC1KDM4ECNR1
SCHEMBL5205241 0.80 KDM4E (0.46) KDM4ETAAR1SMN1; SMN2CNR1
SCHEMBL5208677 0.80 NR3C1 (0.41) HDAC1KDM4EHIF1ATAAR1SMN1; SMN2
SCHEMBL6177393 0.79 ADAMTS5 (0.38) HDAC1ADAMTS5PTGDR2
SCHEMBL6186419 0.79 HDAC1 (0.43) HDAC1KDM4EADAMTS5TAAR1CNR1
SCHEMBL5202191 0.78 PPARG (0.42) SMN1; SMN2PTGDR2FFAR1
SCHEMBL6177750 0.78 ADAMTS5 (0.44) ADAMTS5SMN1; SMN2PTGDR2FFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7160887-B1 Aromatic amine derivatives, their production and use TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-01-09 US disclosed
EP-1123918-B1 AROMATIC AMINE DERIVATIVES, PROCESS FOR THE PREPARATION THEREOF AND AGENTS CONTAINING THE SAME TAKEDA PHARMACEUTICAL (JP) 2005-03-09 EP disclosed
EP-1123918-A1 AROMATIC AMINE DERIVATIVES, PROCESS FOR THE PREPARATION THEREOF AND AGENTS CONTAINING THE SAME Takeda Chemical Industries, Ltd. (JP) 2001-08-16 EP disclosed